171
TITLE: Development of Blood-Brain Barrier Permeable Nitrocatechol-Based Catechol O-Methyltransferase Inhibitors with Reduced Potential for Hepatotoxicity  Full Text
AUTHORS: Tiago Silva; Tarek Mohamed; Arash Shakeri; Praveen P N Rao; Loreto Martinez Gonzalez; Daniel I Perez; Ana Martinez; Maria Joao Valente; Jorge Garrido; Eugenio Uriarte; Paula Serrao ; Patricio Soares da Silva; Fernando Remiao ; Fernanda Borges ;
PUBLISHED: 2016, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 59, ISSUE: 16
INDEXED IN: Scopus WOS CrossRef: 37
IN MY: ORCID
172
TITLE: Discovery of neurotrophic agents based on hydroxycinnamic acid scaffold  Full Text
AUTHORS: Razieh Hosseini; Fatemeh Moosavi; Hamid Rajaian; Tiago Silva; Diogo M E Magalhaes e Silva; Pedro Soares ; Luciano Saso; Najmeh Edraki; Ramin Miri; Fernanda Borges ; Omidreza Firuzi;
PUBLISHED: 2016, SOURCE: CHEMICAL BIOLOGY & DRUG DESIGN, VOLUME: 88, ISSUE: 6
INDEXED IN: Scopus WOS CrossRef: 13
IN MY: ORCID
173
TITLE: Discovery of the first A(1) adenosine receptor ligand based on the chromone scaffold
AUTHORS: Cagide, F ; Reis, J; Alexandra Gaspar ; Chavarria, D ; Kachler, S; Klotz, KN; Gomes, LR ; Low, JN; Vilar, S; Hripcsak, G; Borges, F ;
PUBLISHED: 2016, SOURCE: RSC ADVANCES, VOLUME: 6, ISSUE: 52
INDEXED IN: Scopus WOS CrossRef: 4
IN MY: ORCID
174
175
TITLE: Evaluation of Antioxidant and Antitrypanosomal Properties of a Selected Series of Synthetic 3-Carboxamidocoumarins
AUTHORS: Munoz, A; Fonseca, A; Matos, MJ ; Uriarte, E; Santana, L; Borges, F ; Figueroa, R; Azar, CO;
PUBLISHED: 2016, SOURCE: CHEMISTRYSELECT, VOLUME: 1, ISSUE: 15
INDEXED IN: Scopus WOS CrossRef: 5
176
TITLE: Exploring coumarin potentialities: development of new enzymatic inhibitors based on the 6-methyl-3-carboxamidocoumarin scaffold
AUTHORS: Fonseca, A; Matos, MJ ; Reis, J; Duarte, Y; Gutierrez, M; Santana, L; Uriarte, E; Borges, F ;
PUBLISHED: 2016, SOURCE: RSC ADVANCES, VOLUME: 6, ISSUE: 55
INDEXED IN: Scopus WOS CrossRef: 13
IN MY: ORCID
177
TITLE: In vitro cellular and mitochondrial toxicity of tolcapone and related nitrocatechols  Full Text
AUTHORS: Silva, T; Simoes, RF; Sardao, V; Oliveira, PJ; Valente, MJ; Silva, R; Remiao, F ; Borges, F ;
PUBLISHED: 2016, SOURCE: 52nd Congress of the European-Societies-of-Toxicology (EUROTOX) in TOXICOLOGY LETTERS, VOLUME: 258
INDEXED IN: WOS CrossRef
IN MY: ORCID
178
TITLE: Lessons from black pepper: piperine and derivatives thereof
AUTHORS: Chavarria, D ; Silva, T; Magalhaes e Silva, DME; Remiao, F ; Borges, F ;
PUBLISHED: 2016, SOURCE: EXPERT OPINION ON THERAPEUTIC PATENTS, VOLUME: 26, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef: 45
IN MY: ORCID
179
TITLE: Ligand-Based Virtual Screening Using Tailored Ensembles: A Prioritization Tool for Dual A(2A) Adenosine Receptor Antagonists/Monoamine Oxidase B Inhibitors
AUTHORS: Aliuska M Morales Helguera; Yunierkis Perez Castillo; Natalia N D S Cordeiro ; Eduardo Tejera; Cesar Paz y Mino; Aminael Sanchez Rodriguez; Marta Teijeira; Evys Ancede Gallardo; Fernando Cagide ; Fernanda Borges ; Maykel Cruz Monteagudo;
PUBLISHED: 2016, SOURCE: CURRENT PHARMACEUTICAL DESIGN, VOLUME: 22, ISSUE: 21
INDEXED IN: Scopus WOS CrossRef: 11
IN MY: ORCID
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