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TITLE: Cellular and Mitochondrial Toxicity of Tolcapone, Entacapone, and New Nitrocatechol Derivatives
AUTHORS: Pinto, Miguel ; Silva, Tiago Barros; Sardao, Vilma A.; Simoes, Rui; Albuquerque, Barbara; Oliveira, Paulo J.; Valente, Maria Joao; Remiao, Fernando ; Soares da Silva, Patricio; Fernandes, Carlos ; Borges, Fernanda ;
PUBLISHED: 2024, SOURCE: ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE, VOLUME: 7, ISSUE: 5
INDEXED IN: Scopus WOS CrossRef: 8 Unpaywall
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TITLE: Decreasing the burden of non-alcoholic fatty liver disease: From therapeutic targets to drug discovery opportunities  Full Text
AUTHORS: Ricardo Amorim; Pedro Soares ; Daniel Chavarria ; Sofia Benfeito ; Fernando Cagide ; José Teixeira ; Paulo Oliveira; Fernanda Borges ;
PUBLISHED: 2024, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 277
INDEXED IN: Scopus WOS CrossRef: 9 Unpaywall
13
TITLE: Discovery of a Potent, Selective, and Blood-Brain Barrier Permeable Non-nitrocatechol Inhibitor of Catechol-<i>O</i>-methyltransferase  Full Text
AUTHORS: Benfeito, Sofia ; Albuquerque, Barbara; Sequeira, Lisa ; Lima, Carla; Chavarria, Daniel; Serrao, Paula ; Cagide, Fernando ; Soares da Silva, Patriicio; Borges, Fernanda ;
PUBLISHED: 2024, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 67, ISSUE: 20
INDEXED IN: Scopus WOS CrossRef: 3 Unpaywall
14
TITLE: Drug Development for Alzheimer's and Parkinson's Disease: Where Do We Go Now?  Full Text
AUTHORS: Sequeira, Lisa ; Benfeito, Sofia ; Fernandes, Carlos ; Lima, Ines; Peixoto, Joana; Alves, Catarina; Machado, Claudia Sofia; Alexandra Gaspar ; Borges, Fernanda ; Chavarria, Daniel ;
PUBLISHED: 2024, SOURCE: PHARMACEUTICS, VOLUME: 16, ISSUE: 6
INDEXED IN: Scopus WOS CrossRef: 13 Unpaywall
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TITLE: Dual action of benzaldehydes: Inhibiting quorum sensing and enhancing antibiotic efficacy for controlling Pseudomonas aeruginosa biofilms  Full Text
AUTHORS: Leitao, Miguel M.; Vieira, Tatiana F.; Sousa, Sergio F.; Borges, Fernanda ; Simoes, Manuel ; Borges, Anabela ;
PUBLISHED: 2024, SOURCE: MICROBIAL PATHOGENESIS, VOLUME: 191
INDEXED IN: Scopus WOS CrossRef: 11 Unpaywall
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TITLE: Dual Inhibitors of Brain Carbonic Anhydrases and Monoamine Oxidase-B Efficiently Protect against Amyloid-β-Induced Neuronal Toxicity, Oxidative Stress, and Mitochondrial Dysfunction  Full Text
AUTHORS: Carradori, Simone; Chavarria, Daniel ; Provensi, Gustavo; Leri, Manuela; Bucciantini, Monica; Carradori, Simone; Bonardi, Alessandro; Gratteri, Paola; Borges, Fernanda ; Nocentini, Alessio; Supuran, Claudiu T.;
PUBLISHED: 2024, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 67, ISSUE: 5
INDEXED IN: Scopus WOS CrossRef: 22 Unpaywall
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TITLE: Exploring Nanocarriers for Boosting Entacapone Bioavailability: A Journey through System Characterization and Assessment of Toxicity and Pharmacological and 2D Permeability Paybacks
AUTHORS: Machado, Claudia Sofia; Pinto, Miguel; Aguiar, Brandon; Costa, Sofia; Sarmento, Bruno ; Otero Espinar, Francisco J.; Borges, Fernanda ; Fernandes, Carlos ;
PUBLISHED: 2024, SOURCE: ACS APPLIED MATERIALS & INTERFACES, VOLUME: 16, ISSUE: 43
INDEXED IN: Scopus WOS CrossRef: 5
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TITLE: Insights into the mechanistic pathways underlying the neurotoxic effects of 2C-I and 25I-NBOMe drugs  Full Text
AUTHORS: Gil Martins, E.; Cagide, F. ; Borer, A.; Barbosa, D. J.; Fernandes, C. ; Remiao, F. ; Borges, F. ; Silva, R.;
PUBLISHED: 2024, SOURCE: TOXICOLOGY LETTERS, VOLUME: 399
INDEXED IN: WOS CrossRef
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TITLE: Mechanistic Insights into the Neurotoxicity of 2,5-Dimethoxyphenethylamines (2C) and Corresponding N-(2-methoxybenzyl)phenethylamine (NBOMe) Drugs  Full Text
AUTHORS: Gil Martins, Eva; Cagide Fagin, Fernando ; Martins, Daniel; Borer, Ana; Barbosa, Daniel Jose; Fernandes, Carlos ; Chavarria, Daniel ; Remiao, Fernando ; Borges, Fernanda ; Silva, Renata;
PUBLISHED: 2024, SOURCE: JOURNAL OF XENOBIOTICS, VOLUME: 14, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef: 2 Unpaywall
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