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TITLE: Structural Optimization of Antimycobacterial Azaaurones Towards Improved Solubility and Metabolic Stability  Full Text
AUTHORS: André Campaniço; Shrika Harjivan; Elisabete Freitas; Marco Serafini; Manuela Gaspar ; Rita Capela; Pedro Gomes; Audrey Jordaan; Ana Madureira; Vânia André ; Andreia Silva; Teresa Duarte; Isabel Portugal; João Perdigão; Rui Moreira ; Digby Warner; Francisca Lopes ;
PUBLISHED: 2023, SOURCE: ChemMedChem, VOLUME: 18, ISSUE: 24
INDEXED IN: Scopus CrossRef: 4
13
TITLE: Chemoproteomics-Enabled Identification of 4-Oxo-beta-Lactams as Inhibitors of Dipeptidyl Peptidases 8 and 9
AUTHORS: Carvalho, Luis A. R.; Ross, Breyan; Fehr, Lorenz; Bolgi, Oguz; Woehrle, Svenja; Lum, Kenneth M.; Podlesainski, David; Vieira, Andreia C.; Kiefersauer, Reiner; Felix, Rita; Rodrigues, Tiago; Lucas, Susana D.; Gross, Olaf; Geiss Friedlander, Ruth; Cravatt, Benjamin F.; Huber, Robert; Kaiser, Markus; Moreira, Rui ;
PUBLISHED: 2022, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, VOLUME: 61, ISSUE: 47
INDEXED IN: Scopus WOS CrossRef: 4
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TITLE: Chemoproteomik‐basierte Identifikation von 4‐Oxo‐β‐lactamen als Inhibitoren der Dipeptidylpeptidasen 8 und 9
AUTHORS: Luís A R Carvalho; Breyan Ross; Lorenz Fehr; Oguz Bolgi; Svenja Wöhrle; Kenneth M Lum; David Podlesainski; Andreia C Vieira; Reiner Kiefersauer; Rita Félix; Tiago Rodrigues; Susana D Lucas; Olaf Groß; Ruth Geiss‐Friedlander; Benjamin F Cravatt; Robert Huber; Markus Kaiser; Rui Moreira ;
PUBLISHED: 2022, SOURCE: Angewandte Chemie, VOLUME: 134, ISSUE: 47
INDEXED IN: CrossRef: 1
15
TITLE: Discovery of XL01126: A Potent, Fast, Cooperative, Selective, Orally Bioavailable, and Blood-Brain Barrier Penetrant PROTAC Degrader of Leucine-Rich Repeat Kinase 2
AUTHORS: Liu, Xingui; Kalogeropulou, Alexia F.; Domingos, Sofia; Makukhin, Nikolai; Nirujogi, Raja S.; Singh, Francois; Shpiro, Natalia; Saalfrank, Anton; Sammler, Esther; Ganley, Ian G.; Moreira, Rui ; Alessi, Dario R.; Ciulli, Alessio;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 37
INDEXED IN: Scopus WOS CrossRef: 72
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TITLE: Harnessing Protein-Ligand Interaction Fingerprints to Predict New Scaffolds of RIPK1 Inhibitors  Full Text
AUTHORS: Aniceto, Natalia; Marques, Vanda; Amaral, Joana D.; Serra, Patricia A.; Moreira, Rui ; Rodrigues, Cecilia M. P. ; Guedes, Rita C.;
PUBLISHED: 2022, SOURCE: MOLECULES, VOLUME: 27, ISSUE: 15
INDEXED IN: Scopus WOS CrossRef: 1
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TITLE: Indole-Containing Pyrazino[2,1-b]quinazoline-3,6-diones Active against Plasmodium and Trypanosomatids
AUTHORS: Long, S; Duarte, D; Carvalho, C; Oliveira, R; Santarem, N; Palmeira, A ; Resende, DISP; Silva, AMS; Moreira, R ; Kijjoa, A; da Silva, AC ; Nogueira, F; Sousa, E ; Pinto, MMM;
PUBLISHED: 2022, SOURCE: ACS MEDICINAL CHEMISTRY LETTERS, VOLUME: 13, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef: 4 Unpaywall
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TITLE: Tandem Thio-Michael Addition/Remote Lactone Activation of 5-Hydroxymethylfurfural-Derived delta-Lactone-Fused Cyclopentenones  Full Text
AUTHORS: Gomes, RFA; Ravasco, JMJM; Andrade, KHS; Coelho, JAS; Moreira, R ; Oliveira, R; Nogueira, F; Afonso, CAM;
PUBLISHED: 2022, SOURCE: CHEMSUSCHEM, VOLUME: 15, ISSUE: 13
INDEXED IN: Scopus WOS CrossRef
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TITLE: The Facets of Diversity: The EFMC Perspective
AUTHORS: Borsari, Chiara; Matagne, Brieuc; Goncharenko, Kristina; Moreira, Rui ; Auberson, Yves P.;
PUBLISHED: 2022, SOURCE: CHEMMEDCHEM, VOLUME: 18, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef: 5
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TITLE: Augmenting Adaptive Machine Learning with Kinetic Modeling for Reaction Optimization
AUTHORS: Almeida, AF; Ataide, FAP; Loureiro, RMS; Moreira, R ; Rodrigues, T;
PUBLISHED: 2021, SOURCE: JOURNAL OF ORGANIC CHEMISTRY, VOLUME: 86, ISSUE: 20
INDEXED IN: Scopus WOS CrossRef: 11
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