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TITLE: New azaaurone derivatives as potential multitarget agents in HIV-TB coinfection  Full Text
AUTHORS: Leite, Debora I.; Campanico, Andre; Costa, Pedro A. G.; Correa, Isadora A.; da Costa, Luciana J.; Bastos, Monica M.; Moreira, Rui ; Lopes, Francisca ; Jordaan, Audrey; Warner, Digby F.; Boechat, Nubia;
PUBLISHED: 2023, SOURCE: ARCHIV DER PHARMAZIE, VOLUME: 357, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef: 1
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TITLE: New Compound Combining an Integrase-Targeting Aptamer and a Small Interfering RNA Targeting the Trans-Activation Response/Poly A Region of HIV-1 Potently Suppresses HIV-1 Replication
AUTHORS: Inês Moranguinho; Pedro Borrego ; João Lavrado; Rui Moreira ; Nuno Taveira ;
PUBLISHED: 2023, SOURCE: The 6th International Congress of CiiEM—Immediate and Future Challenges to Foster One Health
INDEXED IN: CrossRef
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TITLE: Structural Optimization of Antimycobacterial Azaaurones Towards Improved Solubility and Metabolic Stability  Full Text
AUTHORS: André Campaniço; Shrika Harjivan; Elisabete Freitas; Marco Serafini; Manuela Gaspar ; Rita Capela; Pedro Gomes; Audrey Jordaan; Ana Madureira; Vânia André ; Andreia Silva; Teresa Duarte; Isabel Portugal; João Perdigão; Rui Moreira ; Digby Warner; Francisca Lopes ;
PUBLISHED: 2023, SOURCE: ChemMedChem, VOLUME: 18, ISSUE: 24
INDEXED IN: Scopus CrossRef: 4
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TITLE: Chemoproteomics-Enabled Identification of 4-Oxo-beta-Lactams as Inhibitors of Dipeptidyl Peptidases 8 and 9
AUTHORS: Carvalho, Luis A. R.; Ross, Breyan; Fehr, Lorenz; Bolgi, Oguz; Woehrle, Svenja; Lum, Kenneth M.; Podlesainski, David; Vieira, Andreia C.; Kiefersauer, Reiner; Felix, Rita; Rodrigues, Tiago; Lucas, Susana D.; Gross, Olaf; Geiss Friedlander, Ruth; Cravatt, Benjamin F.; Huber, Robert; Kaiser, Markus; Moreira, Rui ;
PUBLISHED: 2022, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, VOLUME: 61, ISSUE: 47
INDEXED IN: Scopus WOS CrossRef: 4
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TITLE: Chemoproteomik‐basierte Identifikation von 4‐Oxo‐β‐lactamen als Inhibitoren der Dipeptidylpeptidasen 8 und 9
AUTHORS: Luís A R Carvalho; Breyan Ross; Lorenz Fehr; Oguz Bolgi; Svenja Wöhrle; Kenneth M Lum; David Podlesainski; Andreia C Vieira; Reiner Kiefersauer; Rita Félix; Tiago Rodrigues; Susana D Lucas; Olaf Groß; Ruth Geiss‐Friedlander; Benjamin F Cravatt; Robert Huber; Markus Kaiser; Rui Moreira ;
PUBLISHED: 2022, SOURCE: Angewandte Chemie, VOLUME: 134, ISSUE: 47
INDEXED IN: CrossRef: 1
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TITLE: Discovery of XL01126: A Potent, Fast, Cooperative, Selective, Orally Bioavailable, and Blood-Brain Barrier Penetrant PROTAC Degrader of Leucine-Rich Repeat Kinase 2
AUTHORS: Liu, Xingui; Kalogeropulou, Alexia F.; Domingos, Sofia; Makukhin, Nikolai; Nirujogi, Raja S.; Singh, Francois; Shpiro, Natalia; Saalfrank, Anton; Sammler, Esther; Ganley, Ian G.; Moreira, Rui ; Alessi, Dario R.; Ciulli, Alessio;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 37
INDEXED IN: Scopus WOS CrossRef: 72
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TITLE: DOPING POLYSULFONE DIALYSIS MEMBRANES WITH HUMAN NEUTROPHIL ELASTASE INHIBITORS - A PROOF-OF-CONCEPT STUDY
AUTHORS: Rocha, Susana; Rebelo, Rute; Amorim, Celia ; Moreira, Rui ; Alice Santos-Silva ; Da Silva Montenegro, Maria Conceicao Branco;
PUBLISHED: 2022, SOURCE: NEPHROLOGY DIALYSIS TRANSPLANTATION, VOLUME: 37, ISSUE: Supplement_3
INDEXED IN: WOS CrossRef
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TITLE: Harnessing Protein-Ligand Interaction Fingerprints to Predict New Scaffolds of RIPK1 Inhibitors  Full Text
AUTHORS: Aniceto, Natalia; Marques, Vanda; Amaral, Joana D.; Serra, Patricia A.; Moreira, Rui ; Rodrigues, Cecilia M. P. ; Guedes, Rita C.;
PUBLISHED: 2022, SOURCE: MOLECULES, VOLUME: 27, ISSUE: 15
INDEXED IN: Scopus WOS CrossRef: 1
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TITLE: Indole-Containing Pyrazino[2,1-b]quinazoline-3,6-diones Active against Plasmodium and Trypanosomatids
AUTHORS: Long, S; Duarte, D; Carvalho, C; Oliveira, R; Santarem, N; Palmeira, A ; Resende, DISP; Silva, AMS; Moreira, R ; Kijjoa, A; da Silva, AC ; Nogueira, F; Sousa, E ; Pinto, MMM;
PUBLISHED: 2022, SOURCE: ACS MEDICINAL CHEMISTRY LETTERS, VOLUME: 13, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef: 4 Unpaywall
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