21
TITLE: Discovery of XL01126: A Potent, Fast, Cooperative, Selective, Orally Bioavailable, and Blood-Brain Barrier Penetrant PROTAC Degrader of Leucine-Rich Repeat Kinase 2
AUTHORS: Liu, Xingui; Kalogeropulou, Alexia F.; Domingos, Sofia; Makukhin, Nikolai; Nirujogi, Raja S.; Singh, Francois; Shpiro, Natalia; Saalfrank, Anton; Sammler, Esther; Ganley, Ian G.; Moreira, Rui; Alessi, Dario R.; Ciulli, Alessio;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 37
INDEXED IN: Scopus WOS CrossRef: 72
IN MY: ORCID
22
TITLE: Chemoproteomics-Enabled Identification of 4-Oxo-beta-Lactams as Inhibitors of Dipeptidyl Peptidases 8 and 9
AUTHORS: Carvalho, Luis A. R.; Ross, Breyan; Fehr, Lorenz; Bolgi, Oguz; Woehrle, Svenja; Lum, Kenneth M.; Podlesainski, David; Vieira, Andreia C.; Kiefersauer, Reiner; Felix, Rita; Rodrigues, Tiago; Lucas, Susana D.; Gross, Olaf; Geiss Friedlander, Ruth; Cravatt, Benjamin F.; Huber, Robert; Kaiser, Markus; Moreira, Rui;
PUBLISHED: 2022, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, VOLUME: 61, ISSUE: 47
INDEXED IN: Scopus WOS CrossRef: 4
IN MY: ORCID
23
TITLE: The Facets of Diversity: The EFMC Perspective
AUTHORS: Borsari, Chiara; Matagne, Brieuc; Goncharenko, Kristina; Moreira, Rui; Auberson, Yves P.;
PUBLISHED: 2022, SOURCE: CHEMMEDCHEM, VOLUME: 18, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef: 5
IN MY: ORCID
24
TITLE: Chemoproteomik‐basierte Identifikation von 4‐Oxo‐β‐lactamen als Inhibitoren der Dipeptidylpeptidasen 8 und 9
AUTHORS: Luís A R Carvalho; Breyan Ross; Lorenz Fehr; Oguz Bolgi; Svenja Wöhrle; Kenneth M Lum; David Podlesainski; Andreia C Vieira; Reiner Kiefersauer; Rita Félix; Tiago Rodrigues; Susana D Lucas; Olaf Groß; Ruth Geiss‐Friedlander; Benjamin F Cravatt; Robert Huber; Markus Kaiser; Rui Moreira;
PUBLISHED: 2022, SOURCE: Angewandte Chemie, VOLUME: 134, ISSUE: 47
INDEXED IN: CrossRef: 1
IN MY: ORCID
25
TITLE: Discovery of XL01126: A Potent, Fast, Cooperative, Selective, Oral bioavailable and Blood Brain Barrier Penetrant PROTAC Degrader of Leucine Rich Repeat Kinase 2 (LRRK2)
AUTHORS: Xingui Liu; Alexia Kalogeropulou; Sofia Domingos; Nikolai Makukhin; Raja Nirujogi; Francois Singh; Natalia Shpiro; Anton Saalfrank; Esther Sammler; Ian Ganley; Rui Moreira; Dario Alessi; Alessio Ciulli;
PUBLISHED: 2022
INDEXED IN: CrossRef: 1
IN MY: ORCID
26
TITLE: Nanomedicine Interventions in Clinical Trials for the Treatment of Metastatic Breast Cancer
AUTHORS: Moreira, R; Granja, A; Pinheiro, M; Reis, S ;
PUBLISHED: 2021, SOURCE: APPLIED SCIENCES-BASEL, VOLUME: 11, ISSUE: 4
INDEXED IN: Scopus WOS CrossRef
27
TITLE: Recovery of Depleted miR-146a in ALS Cortical Astrocytes Reverts Cell Aberrancies and Prevents Paracrine Pathogenicity on Microglia and Motor Neurons
AUTHORS: Barbosa, M; Gomes, C; Sequeira, C; Goncalves Ribeiro, J; Pina, CC; Carvalho, LA; Moreira, R; Vaz, SH; Vaz, AR; Brites, D;
PUBLISHED: 2021, SOURCE: FRONTIERS IN CELL AND DEVELOPMENTAL BIOLOGY, VOLUME: 09
INDEXED IN: Scopus WOS CrossRef: 28
IN MY: ORCID
28
TITLE: Discovery of a Necroptosis Inhibitor Improving Dopaminergic Neuronal Loss after MPTP Exposure in Mice  Full Text
AUTHORS: Oliveira, SR; Dionisio, PA; Gaspar, MM; Ferreira, MBT; Rodrigues, CAB; Pereira, RG; Estevao, MS; Perry, MJ; Moreira, R; Afonso, CAM; Amaral, JD; Rodrigues, CMP;
PUBLISHED: 2021, SOURCE: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, VOLUME: 22, ISSUE: 10
INDEXED IN: Scopus WOS CrossRef: 8
IN MY: ORCID
29
TITLE: Two kinematic data-based approaches for cane event detection
AUTHORS: Ribeiro, NF; Mouta, P; Santos, CP;
PUBLISHED: 2021, SOURCE: JOURNAL OF AMBIENT INTELLIGENCE AND HUMANIZED COMPUTING
INDEXED IN: Scopus WOS
30
TITLE: Towards the sustainable discovery and development of new antibiotics
AUTHORS: Miethke, M; Pieroni, M; Weber, T; Bronstrup, M; Hammann, P; Halby, L; Arimondo, PB; Glaser, P; Aigle, B; Bode, HB; Moreira, R; Li, YN; Luzhetskyy, A; Medema, MH; Pernodet, JL; Stadler, M; Tormo, JR; Genilloud, O; Truman, AW; Weissman, KJ; Takano, E; Sabatini, S; Stegmann, E; Brotz Oesterhelt, H; Wohlleben, W; Seemann, M; Empting, M; Hirsch, AKH; Loretz, B; Lehr, CM; Titz, A; Herrmann, J; Jaeger, T; Alt, S; Hesterkamp, T; Winterhalter, M; Schiefer, A; Pfarr, K; Hoerauf, A; Graz, H; Graz, M; Lindvall, M; Ramurthy, S; Karlen, A; van Dongen, M; Petkovic, H; Keller, A; Peyrane, F; Donadio, S; Fraisse, L; Piddock, LJV; Gilbert, IH; Moser, HE; Muller, R; ...More
PUBLISHED: 2021, SOURCE: NATURE REVIEWS CHEMISTRY, VOLUME: 5, ISSUE: 10
INDEXED IN: Scopus WOS CrossRef: 520
IN MY: ORCID
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