11
TITLE: Design, synthesis and biological evaluation of antiparasitic dinitroaniline-ether phospholipid hybrids
AUTHORS: Roussaki, Marina; Magoulas, George E.; Fotopoulou, Theano; Santarem, Nuno; Barrias, Emile; Pohner, Ina; Luelmo, Sara; Afroudakis, Pantelis; Georgikopoulou, Kalliopi; Nevado, Paloma Tejera; Eick, Julia; Bifeld, Eugenia; Corral, Maria J.; Jimenez Anton, Maria Dolores; Ellinger, Bernhard; Kuzikov, Maria; Fragiadaki, Irini; Scoulica, Effie; Gul, Sheraz; Clos, Joachim; Prousis, Kyriakos C.; Torrado, Juan J.; Alunda, Jose Maria; Wade, Rebecca C.; de Souza, Wanderley; da Silva, Anabela Cordeiro ; Calogeropoulou, Theodora; ...More
PUBLISHED: 2023, SOURCE: BIOORGANIC CHEMISTRY, VOLUME: 138
INDEXED IN: Scopus WOS CrossRef: 1
IN MY: ORCID
12
TITLE: Synthesis and Evaluation of Marine-Inspired Compounds Result in Hybrids with Antitrypanosomal and Antileishmanial Activities  Full Text
AUTHORS: Carvalho, Diogo Teixeira; Teixeira, Melissa; Luelmo, Sara; Santarem, Nuno; Pinto, Eugenia ; Cordeiro da Silva, Anabela ; Sousa, Emilia ;
PUBLISHED: 2023, SOURCE: MARINE DRUGS, VOLUME: 21, ISSUE: 11
INDEXED IN: Scopus WOS CrossRef
IN MY: ORCID
13
TITLE: High-Throughput Phenotypic Screening and Machine Learning Methods Enabled the Selection of Broad-Spectrum Low-Toxicity Antitrypanosomatidic Agents
AUTHORS: Linciano, Pasquale; Quotadamo, Antonio; Luciani, Rosaria; Santucci, Matteo; Zorn, Kimberley M.; Foil, Daniel H.; Lane, Thomas R.; da Silva, Anabela Cordeiro ; Santarem, Nuno; Moraes, Carolina B.; Freitas Junior, Lucio; Wittig, Ulrike; Mueller, Wolfgang; Tonelli, Michele; Ferrari, Stefania; Venturelli, Alberto; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Reinshagen, Jeanette; Ekins, Sean; Costi, Maria Paola; ...More
PUBLISHED: 2023, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 66, ISSUE: 22
INDEXED IN: Scopus WOS CrossRef: 3
IN MY: ORCID
14
TITLE: Guidelines for the purification and characterization of extracellular vesicles of parasites
AUTHORS: Carmen Fernandez Becerra; Patrícia Xander; Daniel Alfandari; George Dong; Iris Aparici Herraiz; Irit Rosenhek Goldian; Mehrdad Shokouhy; Melisa Gualdron Lopez; Nicholy Lozano; Nuria Cortes Serra; Paula Abou Karam; Paula Meneghetti; Rafael Pedro Madeira; Ziv Porat; Rodrigo Pedro Soares; Adriana Oliveira Costa; Sima Rafati; Anabela Cordeiro da Silva ; Nuno Santarém; Christopher Fernandez Prada; Marcel I Ramirez; Dolores Bernal; Antonio Marcilla; Vera Lucia Pereira Chioccola; Lysangela Ronalte Alves; Hernando Del Portillo; Neta Regev Rudzki; Igor Correia de Almeida; Sergio Schenkman; Martin Olivier; Ana Claudia Torrecilhas; ...More
PUBLISHED: 2023, SOURCE: Journal of Extracellular Biology, VOLUME: 2, ISSUE: 10
INDEXED IN: Scopus CrossRef: 14 Unpaywall
IN MY: ORCID
15
TITLE: Indole-Containing Pyrazino[2,1-b]quinazoline-3,6-diones Active against Plasmodium and Trypanosomatids
AUTHORS: Long, S; Duarte, D; Carvalho, C; Oliveira, R; Santarem, N; Palmeira, A ; Resende, DISP; Silva, AMS; Moreira, R ; Kijjoa, A; da Silva, AC ; Nogueira, F; Sousa, E ; Pinto, MMM;
PUBLISHED: 2022, SOURCE: ACS MEDICINAL CHEMISTRY LETTERS, VOLUME: 13, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef: 4 Unpaywall
IN MY: ORCID
16
TITLE: IgG functionalized polymeric nanoparticles for oral insulin administration  Full Text
AUTHORS: De Marchi, J. G. B.; Ce, R.; Onzi, G.; Alves, A. C. S.; Santarem, N.; Cordeiro da Silva, A. ; Pohlmann, A. R.; Guterres, S. S.; Ribeiro, A. J.;
PUBLISHED: 2022, SOURCE: INTERNATIONAL JOURNAL OF PHARMACEUTICS, VOLUME: 622
INDEXED IN: Scopus WOS CrossRef: 5
IN MY: ORCID
17
TITLE: Current Treatments to Control African Trypanosomiasis and One Health Perspective
AUTHORS: Venturelli, Alberto; Tagliazucchi, Lorenzo; Lima, Clara; Venuti, Federica; Malpezzi, Giulia; Magoulas, George E.; Santarem, Nuno; Calogeropoulou, Theodora; Cordeiro da Silva, Anabela ; Costi, Maria Paola;
PUBLISHED: 2022, SOURCE: MICROORGANISMS, VOLUME: 10, ISSUE: 7
INDEXED IN: Scopus WOS CrossRef: 4
IN MY: ORCID
18
TITLE: Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1  Full Text
AUTHORS: Poehner, Ina; Quotadamo, Antonio; Panecka Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro da Silva, Anabela ; Costi, Maria P.; Venturelli, Alberto; Wade, Rebecca C.;
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 65, ISSUE: 13
INDEXED IN: Scopus WOS CrossRef: 2
IN MY: ORCID
19
TITLE: Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1  Full Text
AUTHORS: Poehner, Ina; Quotadamo, Antonio; Panecka Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro da Silva, Anabela; Costi, Maria P.; Venturelli, Alberto; Wade, Rebecca C.;
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY
INDEXED IN: WOS
20
TITLE: Pyrimido[5,4-d]pyrimidine-Based Compounds as a Novel Class of Antitrypanosomal and Antileishmanial Agents
AUTHORS: Lopes, Andre; Santarem, Nuno; Cordeiro da Silva, Anabela ; Carvalho, M. Alice ;
PUBLISHED: 2022, SOURCE: ACS MEDICINAL CHEMISTRY LETTERS, VOLUME: 13, ISSUE: 9
INDEXED IN: Scopus WOS CrossRef
IN MY: ORCID
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