Goncalo J. L. Bernardes
AuthID: R-00F-QH3
11
TITLE: Ibrutinib Inhibits BMX-Dependent Endothelial VCAM-1 Expression In Vitro and Pro-Atherosclerotic Endothelial Activation and Platelet Adhesion In Vivo Full Text
AUTHORS: Kohs, Tia C. L.; Olson, Sven R.; Pang, Jiaqing; Jordan, Kelley R.; Zheng, Tony J.; Xie, Aris; Hodovan, James; Muller, Matthew; McArthur, Carrie; Johnson, Jennifer; Sousa, Barbara B.; Wallisch, Michael; Kievit, Paul; Aslan, Joseph E.; Seixas, Joao D.; Bernardes, Goncalo J. L.; Hinds, Monica T.; Lindner, Jonathan R.; McCarty, Owen J. T.; Puy, Cristina; ...More
PUBLISHED: 2022, SOURCE: CELLULAR AND MOLECULAR BIOENGINEERING, VOLUME: 15, ISSUE: 3
AUTHORS: Kohs, Tia C. L.; Olson, Sven R.; Pang, Jiaqing; Jordan, Kelley R.; Zheng, Tony J.; Xie, Aris; Hodovan, James; Muller, Matthew; McArthur, Carrie; Johnson, Jennifer; Sousa, Barbara B.; Wallisch, Michael; Kievit, Paul; Aslan, Joseph E.; Seixas, Joao D.; Bernardes, Goncalo J. L.; Hinds, Monica T.; Lindner, Jonathan R.; McCarty, Owen J. T.; Puy, Cristina; ...More
PUBLISHED: 2022, SOURCE: CELLULAR AND MOLECULAR BIOENGINEERING, VOLUME: 15, ISSUE: 3
INDEXED IN:
Scopus
WOS
12
TITLE: Transition metal mediated bioorthogonal release
AUTHORS: Sabatino, Valerio; Unnikrishnan, V. B.; Bernardes, Goncalo J. L.;
PUBLISHED: 2022, SOURCE: CHEM CATALYSIS, VOLUME: 2, ISSUE: 1
AUTHORS: Sabatino, Valerio; Unnikrishnan, V. B.; Bernardes, Goncalo J. L.;
PUBLISHED: 2022, SOURCE: CHEM CATALYSIS, VOLUME: 2, ISSUE: 1
INDEXED IN:
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13
TITLE: Platform for Orthogonal N-Cysteine-Specific Protein Modification Enabled by Cyclopropenone Reagents Full Text
AUTHORS: Istrate, Alena; Geeson, Michael B.; Navo, Claudio D.; Sousa, Barbara B.; Marques, Marta C.; Taylor, Ross J.; Journeaux, Toby; Oehler, Sebastian R.; Mortensen, Michael R.; Deery, Michael J.; Bond, Andrew D.; Corzana, Francisco; Jimenez Oses, Gonzalo; Bernardes, Goncalo J. L.;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 23
AUTHORS: Istrate, Alena; Geeson, Michael B.; Navo, Claudio D.; Sousa, Barbara B.; Marques, Marta C.; Taylor, Ross J.; Journeaux, Toby; Oehler, Sebastian R.; Mortensen, Michael R.; Deery, Michael J.; Bond, Andrew D.; Corzana, Francisco; Jimenez Oses, Gonzalo; Bernardes, Goncalo J. L.;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 23
INDEXED IN:
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14
TITLE: Chemical and Enzymatic Methods for Post-Translational Protein-Protein Conjugation Full Text
AUTHORS: Taylor, Ross J.; Geeson, Michael B.; Journeaux, Toby; Bernardes, Goncalo J. L.;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 32
AUTHORS: Taylor, Ross J.; Geeson, Michael B.; Journeaux, Toby; Bernardes, Goncalo J. L.;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 32
INDEXED IN:
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15
TITLE: Selective Inhibition of Bruton?s Tyrosine Kinase by a Designed Covalent Ligand Leads to Potent Therapeutic Efficacy in Blood Cancers Relative to Clinically Used Inhibitors
AUTHORS: Sousa, Barbara B.; De Almeida, Catia Rebelo; Barahona, Ana F.; Lopes, Raquel; Martins Logrado, Ana; Cavaco, Marco; Neves, Vera; Carvalho, Luis A. R.; Labao Almeida, Carlos; Coelho, Ana R.; Bento, Marta Leal; Lopes, Ricardo M. R. M.; Oliveira, Bruno L.; Castanho, Miguel A. R. B.; Neumeister, Peter; Deutsch, Alexander; Vladimer, Gregory I.; Krall, Nikolaus; Joao, Cristina; Corzana, Francisco; ...More
PUBLISHED: 2022, SOURCE: ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE, VOLUME: 5, ISSUE: 11
AUTHORS: Sousa, Barbara B.; De Almeida, Catia Rebelo; Barahona, Ana F.; Lopes, Raquel; Martins Logrado, Ana; Cavaco, Marco; Neves, Vera; Carvalho, Luis A. R.; Labao Almeida, Carlos; Coelho, Ana R.; Bento, Marta Leal; Lopes, Ricardo M. R. M.; Oliveira, Bruno L.; Castanho, Miguel A. R. B.; Neumeister, Peter; Deutsch, Alexander; Vladimer, Gregory I.; Krall, Nikolaus; Joao, Cristina; Corzana, Francisco; ...More
PUBLISHED: 2022, SOURCE: ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE, VOLUME: 5, ISSUE: 11
INDEXED IN:
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16
TITLE: Facile installation of post-translational modifications on the tau protein via chemical mutagenesis
AUTHORS: Vendruscolo, M; Bernardes, GJL; Lindstedt, PR; Taylor, RJ;
PUBLISHED: 2021, SOURCE: ACS Chemical Neuroscience
AUTHORS: Vendruscolo, M; Bernardes, GJL; Lindstedt, PR; Taylor, RJ;
PUBLISHED: 2021, SOURCE: ACS Chemical Neuroscience
INDEXED IN:
Scopus
17
TITLE: Facile Installation of Post-translational Modifications on the Tau Protein via Chemical Mutagenesis
AUTHORS: Lindstedt, PR; Taylor, RJ; Bernardes, GJL; Vendruscolo, M;
PUBLISHED: 2021, SOURCE: ACS CHEMICAL NEUROSCIENCE, VOLUME: 12, ISSUE: 3
AUTHORS: Lindstedt, PR; Taylor, RJ; Bernardes, GJL; Vendruscolo, M;
PUBLISHED: 2021, SOURCE: ACS CHEMICAL NEUROSCIENCE, VOLUME: 12, ISSUE: 3
INDEXED IN:
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18
TITLE: Precise protein conjugation technology for the construction of homogenous glycovaccines
AUTHORS: Kitowski, A; Corzana, F; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: Drug Discovery Today: Technologies
AUTHORS: Kitowski, A; Corzana, F; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: Drug Discovery Today: Technologies
INDEXED IN:
Scopus
19
TITLE: The role of reversible and irreversible covalent chemistry in targeted protein degradation
AUTHORS: Kiely Collins, H; Winter, GE; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: CELL CHEMICAL BIOLOGY, VOLUME: 28, ISSUE: 7
AUTHORS: Kiely Collins, H; Winter, GE; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: CELL CHEMICAL BIOLOGY, VOLUME: 28, ISSUE: 7
INDEXED IN:
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20
TITLE: Exploration of Long-Chain Vitamin E Metabolites for the Discovery of a Highly Potent, Orally Effective, and Metabolically Stable 5-LOX Inhibitor that Limits Inflammation Full Text
AUTHORS: Neukirch, K; Alsabil, K; Dinh, CP; Bilancia, R; Raasch, M; Ville, A; Cerqua, I; Viault, G; Breard, D; Pace, S; Temml, V; Brunner, E; Jordan, PM; Marques, MC; Loeser, K; Gollowitzer, A; Permann, S; Gerstmeier, J; Lorkowski, S; Stuppner, H; ...More
PUBLISHED: 2021, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 64, ISSUE: 15
AUTHORS: Neukirch, K; Alsabil, K; Dinh, CP; Bilancia, R; Raasch, M; Ville, A; Cerqua, I; Viault, G; Breard, D; Pace, S; Temml, V; Brunner, E; Jordan, PM; Marques, MC; Loeser, K; Gollowitzer, A; Permann, S; Gerstmeier, J; Lorkowski, S; Stuppner, H; ...More
PUBLISHED: 2021, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 64, ISSUE: 15
INDEXED IN:
Scopus
WOS