21
TITLE: Chemical and Enzymatic Methods for Post-Translational Protein-Protein Conjugation  Full Text
AUTHORS: Taylor, Ross J.; Geeson, Michael B.; Journeaux, Toby; Bernardes, Goncalo J. L.;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 32
INDEXED IN: Scopus WOS
22
TITLE: Cysteine-Assisted Click-Chemistry for Proximity-Driven, Site-Specific Acetylation of Histones  Full Text
AUTHORS: Afonso, Claudia F.; Marques, Marta C.; Antonio, Joao P. M.; Cordeiro, Carlos; Gois, Pedro M. P.; Cal, Pedro M. S. D.; Bernardes, Goncalo J. L.;
PUBLISHED: 2022, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
INDEXED IN: Scopus WOS
23
TITLE: Selective Inhibition of Bruton?s Tyrosine Kinase by a Designed Covalent Ligand Leads to Potent Therapeutic Efficacy in Blood Cancers Relative to Clinically Used Inhibitors
AUTHORS: Sousa, Barbara B.; De Almeida, Catia Rebelo; Barahona, Ana F.; Lopes, Raquel; Martins Logrado, Ana; Cavaco, Marco; Neves, Vera; Carvalho, Luis A. R.; Labao Almeida, Carlos; Coelho, Ana R.; Bento, Marta Leal; Lopes, Ricardo M. R. M.; Oliveira, Bruno L.; Castanho, Miguel A. R. B.; Neumeister, Peter; Deutsch, Alexander; Vladimer, Gregory I.; Krall, Nikolaus; Joao, Cristina; Corzana, Francisco; Seixas, Joao D.; Fior, Rita; Bernardes, Goncalo J. L.; ...More
PUBLISHED: 2022, SOURCE: ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE, VOLUME: 5, ISSUE: 11
INDEXED IN: Scopus WOS
24
TITLE: Systematic Activity Maturation of a Single-Domain Antibody with Non-canonical Amino Acids through Chemical Mutagenesis
AUTHORS: Lindstedt, PR; Aprile, FA; Sormanni, P; Rakoto, R; Dobson, CM; Bernardes, GJL; Vendruscolo, M;
PUBLISHED: 2021, SOURCE: CELL CHEMICAL BIOLOGY, VOLUME: 28, ISSUE: 1
INDEXED IN: Scopus WOS
25
TITLE: In Vivo Pretargeting Based on Cysteine-Selective Antibody Modification with IEDDA Bioorthogonal Handles for Click Chemistry  Full Text
AUTHORS: Ferreira, VFC; Oliveira, BL; D'Onofrio, A; Farinha, CM; Gano, L; Paulo, A; Bernardes, GJL; Mendes, F;
PUBLISHED: 2021, SOURCE: BIOCONJUGATE CHEMISTRY, VOLUME: 32, ISSUE: 1
INDEXED IN: Scopus WOS
26
TITLE: Facile installation of post-translational modifications on the tau protein via chemical mutagenesis
AUTHORS: Vendruscolo, M; Bernardes, GJL; Lindstedt, PR; Taylor, RJ;
PUBLISHED: 2021, SOURCE: ACS Chemical Neuroscience
INDEXED IN: Scopus
27
TITLE: Facile Installation of Post-translational Modifications on the Tau Protein via Chemical Mutagenesis
AUTHORS: Lindstedt, PR; Taylor, RJ; Bernardes, GJL; Vendruscolo, M;
PUBLISHED: 2021, SOURCE: ACS CHEMICAL NEUROSCIENCE, VOLUME: 12, ISSUE: 3
INDEXED IN: WOS
28
TITLE: Precise protein conjugation technology for the construction of homogenous glycovaccines
AUTHORS: Kitowski, A; Corzana, F; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: Drug Discovery Today: Technologies
INDEXED IN: Scopus
29
TITLE: The role of reversible and irreversible covalent chemistry in targeted protein degradation
AUTHORS: Kiely Collins, H; Winter, GE; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: CELL CHEMICAL BIOLOGY, VOLUME: 28, ISSUE: 7
INDEXED IN: Scopus WOS
30
TITLE: Allosteric Antagonist Modulation of TRPV2 by Piperlongumine Impairs Glioblastoma Progression
AUTHORS: Conde, J; Pumroy, RA; Baker, C; Rodrigues, T; Guerreiro, A; Sousa, BB; Marques, MC; de Almeida, BP; Lee, S; Leites, EP; Picard, D; Samanta, A; Vaz, SH; Sieglitz, F; Langini, M; Remke, M; Roque, R; Weiss, T; Weller, M; Liu, YH; Han, S; Corzana, F; Morais, VA; Faria, CC; Carvalho, T; Filippakopoulos, P; Snijder, B; Barbosa Morais, NL; Moiseenkova Bell, VY; Bernardes, GJL; ...More
PUBLISHED: 2021, SOURCE: ACS CENTRAL SCIENCE, VOLUME: 7, ISSUE: 5
INDEXED IN: Scopus WOS
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