Goncalo J. L. Bernardes
AuthID: R-00F-QH3
31
TITLE: Protein Conjugation by Electrophilic Alkynylation Using 5-(Alkynyl)dibenzothiophenium Triflates Full Text
AUTHORS: Laserna, V; Istrate, A; Kafuta, K; Hakala, TA; Knowles, TPJ; Alcarazo, M; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: BIOCONJUGATE CHEMISTRY, VOLUME: 32, ISSUE: 8
AUTHORS: Laserna, V; Istrate, A; Kafuta, K; Hakala, TA; Knowles, TPJ; Alcarazo, M; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: BIOCONJUGATE CHEMISTRY, VOLUME: 32, ISSUE: 8
INDEXED IN: 
Scopus 
WOS
Scopus WOS32
TITLE: Arylethynyltrifluoroborate Dienophiles for on Demand Activation of IEDDA Reactions Full Text
AUTHORS: Zawada, Z; Guo, ZJ; Oliveira, BL; Navo, CD; Li, H; Cal, PMSD; Corzana, F; Jimenez Oses, G; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: BIOCONJUGATE CHEMISTRY, VOLUME: 32, ISSUE: 8
AUTHORS: Zawada, Z; Guo, ZJ; Oliveira, BL; Navo, CD; Li, H; Cal, PMSD; Corzana, F; Jimenez Oses, G; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: BIOCONJUGATE CHEMISTRY, VOLUME: 32, ISSUE: 8
INDEXED IN: Scopus WOS
Scopus WOS33
TITLE: Exploration of Long-Chain Vitamin E Metabolites for the Discovery of a Highly Potent, Orally Effective, and Metabolically Stable 5-LOX Inhibitor that Limits Inflammation Full Text
AUTHORS: Neukirch, K; Alsabil, K; Dinh, CP; Bilancia, R; Raasch, M; Ville, A; Cerqua, I; Viault, G; Breard, D; Pace, S; Temml, V; Brunner, E; Jordan, PM; Marques, MC; Loeser, K; Gollowitzer, A; Permann, S; Gerstmeier, J; Lorkowski, S; Stuppner, H; ...More
PUBLISHED: 2021, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 64, ISSUE: 15
AUTHORS: Neukirch, K; Alsabil, K; Dinh, CP; Bilancia, R; Raasch, M; Ville, A; Cerqua, I; Viault, G; Breard, D; Pace, S; Temml, V; Brunner, E; Jordan, PM; Marques, MC; Loeser, K; Gollowitzer, A; Permann, S; Gerstmeier, J; Lorkowski, S; Stuppner, H; ...More
PUBLISHED: 2021, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 64, ISSUE: 15
INDEXED IN: Scopus WOS
Scopus WOS34
TITLE: Dichloro Butenediamides as Irreversible Site-Selective Protein Conjugation Reagent Full Text
AUTHORS: Laserna, V; Abegg, D; Afonso, CF; Martin, EM; Adibekian, A; Ravn, P; Corzana, F; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
AUTHORS: Laserna, V; Abegg, D; Afonso, CF; Martin, EM; Adibekian, A; Ravn, P; Corzana, F; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
INDEXED IN: Scopus WOS
Scopus WOS35
TITLE: Combating small-molecule aggregation with machine learning
AUTHORS: Lee, K; Yang, A; Lin, YC; Reker, D; Bernardes, GJL; Rodrigues, T;
PUBLISHED: 2021, SOURCE: CELL REPORTS PHYSICAL SCIENCE, VOLUME: 2, ISSUE: 9
AUTHORS: Lee, K; Yang, A; Lin, YC; Reker, D; Bernardes, GJL; Rodrigues, T;
PUBLISHED: 2021, SOURCE: CELL REPORTS PHYSICAL SCIENCE, VOLUME: 2, ISSUE: 9
INDEXED IN: Scopus WOS
Scopus WOS36
TITLE: A Platform for Site-Specific DNA-Antibody Bioconjugation by Using Benzoylacrylic-Labelled Oligonucleotides Full Text
AUTHORS: Konc, J; Brown, L; Whiten, DR; Zuo, YK; Ravn, P; Klenerman, D; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
AUTHORS: Konc, J; Brown, L; Whiten, DR; Zuo, YK; Ravn, P; Klenerman, D; Bernardes, GJL;
PUBLISHED: 2021, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
INDEXED IN: WOS
WOS37
TITLE: Diazaborines Are a Versatile Platform to Develop ROS-Responsive Antibody Drug Conjugates** Full Text
AUTHORS: Antonio, JPM; Carvalho, JI; Andre, AS; Dias, JNR; Aguiar, SI; Faustino, H; Lopes, RMRM; Veiros, LF; Bernardes, GJL; Silva, FA; Gois, PMP;
PUBLISHED: 2021, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
AUTHORS: Antonio, JPM; Carvalho, JI; Andre, AS; Dias, JNR; Aguiar, SI; Faustino, H; Lopes, RMRM; Veiros, LF; Bernardes, GJL; Silva, FA; Gois, PMP;
PUBLISHED: 2021, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
INDEXED IN: WOS
WOS38
TITLE: A Structural Ensemble of a Tau-Microtubule Complex Reveals Regulatory Tau Phosphorylation and Acetylation Mechanisms
AUTHORS: Brotzakis, ZF; Lindstedt, PR; Taylor, RJ; Rinauro, DJ; Gallagher, NCT; Bernardes, GJL; Vendruscolo, M;
PUBLISHED: 2021, SOURCE: ACS CENTRAL SCIENCE
AUTHORS: Brotzakis, ZF; Lindstedt, PR; Taylor, RJ; Rinauro, DJ; Gallagher, NCT; Bernardes, GJL; Vendruscolo, M;
PUBLISHED: 2021, SOURCE: ACS CENTRAL SCIENCE
INDEXED IN: Scopus WOS
Scopus WOS39
TITLE: Machine learning for target discovery in drug development Full Text
AUTHORS: Tiago Rodrigues; Goncalo J L Bernardes;
PUBLISHED: 2020, SOURCE: CURRENT OPINION IN CHEMICAL BIOLOGY, VOLUME: 56
AUTHORS: Tiago Rodrigues; Goncalo J L Bernardes;
PUBLISHED: 2020, SOURCE: CURRENT OPINION IN CHEMICAL BIOLOGY, VOLUME: 56
INDEXED IN: Scopus WOS
Scopus WOS40
TITLE: Proteome-Wide Survey of Cysteine Oxidation by Using a Norbornene Probe Full Text
AUTHORS: Lisa J Alcock; Maike Langini; Kai Stuehler; Marc Remke; Michael V Perkins; Goncalo J L Bernardes; Justin M Chalker;
PUBLISHED: 2020, SOURCE: CHEMBIOCHEM, VOLUME: 21, ISSUE: 9
AUTHORS: Lisa J Alcock; Maike Langini; Kai Stuehler; Marc Remke; Michael V Perkins; Goncalo J L Bernardes; Justin M Chalker;
PUBLISHED: 2020, SOURCE: CHEMBIOCHEM, VOLUME: 21, ISSUE: 9
INDEXED IN: Scopus WOS
Scopus WOS