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TITLE: Exploiting the 2-Amino-1,3,4-thiadiazole Scaffold To Inhibit Trypanosoma brucei Pteridine Reductase in Support of Early-Stage Drug Discovery
AUTHORS: Linciano, P; Dawson, A; Pohner, I; Costa, DM; Sa, MS; Cordeiro da Silva, A ; Luciani, R; Gul, S; Witt, G; Ellinger, B; Kuzikov, M; Gribbon, P; Reinshagen, J; Wolf, M; Behrens, B; Hannaert, V; Michels, PAM; Nerini, E; Pozzi, C; di Pisa, F; Landi, G; Santarem, N; Ferrari, S; Saxena, P; Lazzari, S; Cannazza, G; Freitas, LH; Moraes, CB; Pascoalino, BS; Alcantara, LM; Bertolacini, CP; Fontana, V; Wittig, U; Muller, W; Wade, RC; Hunter, WN; Mangani, S; Costantino, L; Costi, MP; ...More
PUBLISHED: 2017, SOURCE: ACS OMEGA, VOLUME: 2, ISSUE: 9
INDEXED IN: Scopus WOS CrossRef: 1
12
TITLE: Profiling of Flavonol Derivatives for the Development of Antitrypanosomatidic Drugs  Full Text
AUTHORS: Chiara Borsari; Rosaria Luciani; Cecilia Pozzi; Ina Poehner; Stefan Henrich; Matteo Trande; Anabela Cordeiro da Silva ; Nuno Santarem; Catarina Baptista; Annalisa Tait; Flavio Di Pisa; Lucia Dello Iacono; Giacomo Landi; Sheraz Gul; Markus Wolf; Maria Kuzikov; Bernhard Ellinger; Jeanette Reinshagen; Gesa Witt; Philip Gribbon; Manfred Kohler; Oliver Keminer; Birte Behrens; Luca Costantino; Paloma Tejera Nevado; Eugenia Bifeld; Julia Eick; Joachim Clos; Juan Torrado; Maria D Jimenez Anton; Maria J Corral; Jose M Ma Alunda; Federica Pellati; Rebecca C Wade; Stefania Ferrari; Stefano Mangani; Maria Paola Costi; ...More
PUBLISHED: 2016, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 59, ISSUE: 16
INDEXED IN: Scopus WOS CrossRef
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