21
TITLE: Deep generative model for therapeutic targets using transcriptomic disease-associated data-USP7 case study
AUTHORS: Pereira, Tiago; Abbasi, Maryam; Oliveira, Rita, I; Guedes, Romina A.; Salvador, Jorge A. R.; Arrais, Joel P.;
PUBLISHED: 2022, SOURCE: BRIEFINGS IN BIOINFORMATICS, VOLUME: 23, ISSUE: 4
INDEXED IN: Scopus WOS CrossRef: 7
IN MY: ORCID
22
TITLE: Therapeutic targeting of PD-1/PD-L1 blockade by novel small-molecule inhibitors recruits cytotoxic T cells into solid tumor microenvironment
AUTHORS: Rita C Acúrcio; Sabina Pozzi; Barbara Carreira; Marta Pojo; Nuria Gómez Cebrián; Sandra Casimiro; Adelaide Fernandes; Andreia Barateiro; Vitor Farricha; Joaquim Brito; Ana Paula Leandro ; Jorge A R Salvador; Luís Graça ; Leonor Puchades Carrasco; Luís Costa; Ronit Satchi Fainaro; Rita C Guedes; Helena F Florindo;
PUBLISHED: 2022, SOURCE: Journal for immunotherapy of cancer, VOLUME: 10, ISSUE: 7
INDEXED IN: Scopus CrossRef: 23
IN MY: ORCID
23
TITLE: Highlights in USP7 inhibitors for cancer treatment
AUTHORS: Oliveira, Rita I.; Guedes, Romina A.; Salvador, Jorge A. R.;
PUBLISHED: 2022, SOURCE: FRONTIERS IN CHEMISTRY, VOLUME: 10
INDEXED IN: Scopus WOS CrossRef: 18
IN MY: ORCID
24
TITLE: MDM2-Based Proteolysis-Targeting Chimeras (PROTACs): An Innovative Drug Strategy for Cancer Treatment
AUTHORS: Vicente, Andre T. S.; Salvador, Jorge A. R.;
PUBLISHED: 2022, SOURCE: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, VOLUME: 23, ISSUE: 19
INDEXED IN: Scopus WOS CrossRef: 17
IN MY: ORCID
25
TITLE: Design, synthesis, and biological evaluation of new arjunolic acid derivatives as anticancer agents
AUTHORS: Gonçalves, BMF; Mendes, VIS; Silvestre, SM; Salvador, JAR;
PUBLISHED: 2022, SOURCE: RSC Medicinal Chemistry, VOLUME: 14, ISSUE: 2
INDEXED IN: Scopus CrossRef: 1
IN MY: ORCID
26
TITLE: Editorial: Head & Neck Cancer and Esophageal Cancer: From Biosignatures to Therapeutics  Full Text
AUTHORS: Kok, VC; Yu, CC; Salvador, JAR;
PUBLISHED: 2021, SOURCE: FRONTIERS IN ONCOLOGY, VOLUME: 11
INDEXED IN: Scopus WOS
27
TITLE: A patent review of glutaminyl cyclase inhibitors (2004-present)
AUTHORS: Coimbra, JRM; Salvador, JAR;
PUBLISHED: 2021, SOURCE: EXPERT OPINION ON THERAPEUTIC PATENTS, VOLUME: 31, ISSUE: 9
INDEXED IN: WOS CrossRef: 8
IN MY: ORCID
28
TITLE: Combining Virtual Screening Protocol and In Vitro Evaluation towards the Discovery of BACE1 Inhibitors  Full Text
AUTHORS: Coimbra, JRM; Baptista, SJ; Dinis, TCP; Silva, MMC; Moreira, PI; Moreira, Paula Isabel; Paula I. Moreira ; Santos, AE; Salvador, JAR;
PUBLISHED: 2020, SOURCE: BIOMOLECULES, VOLUME: 10, ISSUE: 4
INDEXED IN: Scopus WOS CrossRef: 13
IN MY: ORCID
29
TITLE: Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-7  Full Text
AUTHORS: Gutschow, M; Vanden Eynde, JJ; Jampilek, J; Kang, CB; Mangoni, AA; Fossa, P; Karaman, R; Trabocchi, A; Scott, PJH; Reynisson, J; Rapposelli, S; Galdiero, S; Winum, JY; Brullo, C; Prokai Tatrai, K; Sharma, AK; Schapira, M; Azuma, YT; Cerchia, L; Spetea, M; Torri, G; Collina, S; Geronikaki, A; Garcia Sosa, AT; Vasconcelos, MH ; Sousa, ME ; Kosalec, I; Tuccinardi, T; Duarte, IF; Salvador, JAR; Bertinaria, M; Pellecchia, M; Amato, J; Rastelli, G; Paula Gomes ; Guedes, RC; Sabatier, JM; Estevez Braun, A; Pagano, B; Mangani, S; Ragno, R; Kokotos, G; Brindisi, M; Gonzalez, FV; Borges, F ; Miloso, M; Rautio, J; Munoz Torrero, D; ...More
PUBLISHED: 2020, SOURCE: MOLECULES, VOLUME: 25, ISSUE: 13
INDEXED IN: Scopus WOS CrossRef: 5 Unpaywall
IN MY: ORCID
30
TITLE: New BACE1 Chimeric Peptide Inhibitors Selectively Prevent A beta PP-beta Cleavage Decreasing Amyloid-beta Production and Accumulation in Alzheimer's Disease Models
AUTHORS: Resende, R; Ferreira Marques, M; Moreira, P ; Coimbra, JRM; Baptista, SJ; Isidoro, C; Salvador, JAR; Dinis, TCP; Pereira, CF; Santos, AE;
PUBLISHED: 2020, SOURCE: JOURNAL OF ALZHEIMERS DISEASE, VOLUME: 76, ISSUE: 4
INDEXED IN: Scopus WOS CrossRef: 8
IN MY: ORCID
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