1
TITLE: Synthesis, Biological Evaluation, and Docking Studies of Open-Chain Carbohydrate Amides as Acetylcholinesterase Inhibitors
AUTHORS: Goncalves Pereira, Rita; Figueiredo, Jose A.; Lucas, Susana D.; Garcia Moreno, Maria I.; Mellet, Carmen O.; Rauter, Amelia P.; Ismael, Maria I.;
PUBLISHED: 2023, SOURCE: MEDICINAL CHEMISTRY, VOLUME: 19, ISSUE: 6
INDEXED IN: Scopus WOS
2
TITLE: Chemoproteomics-Enabled Identification of 4-Oxo-beta-Lactams as Inhibitors of Dipeptidyl Peptidases 8 and 9  Full Text
AUTHORS: Carvalho, Luis A. R.; Ross, Breyan; Fehr, Lorenz; Bolgi, Oguz; Woehrle, Svenja; Lum, Kenneth M.; Podlesainski, David; Vieira, Andreia C.; Kiefersauer, Reiner; Felix, Rita; Rodrigues, Tiago; Lucas, Susana D.; Gross, Olaf; Geiss Friedlander, Ruth; Cravatt, Benjamin F.; Huber, Robert; Kaiser, Markus; Moreira, Rui;
PUBLISHED: 2022, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION
INDEXED IN: Scopus WOS
5
TITLE: Ursolic and oleanolic acid derivatives with cholinesterase inhibiting potential  Full Text
AUTHORS: Anne Loesche; Alexander Koewitsch; Susana D Lucas; Zayan Al Halabi; Wolfgang Sippl; Ahmed Al Harrasi; Rene Csuk;
PUBLISHED: 2019, SOURCE: BIOORGANIC CHEMISTRY, VOLUME: 85
INDEXED IN: WOS
6
TITLE: Acetylcholinesterase Choline-Based Ionic Liquid Inhibitors: In Vitro and in Silico Molecular Docking Studies
AUTHORS: Siopa, F; Frade, RFM; Diniz, A; Andrade, JM; Nicolai, M; Meirinhos, A; Lucas, SD; Marcelo, F; Afonso, CAM; Rijo, P ;
PUBLISHED: 2018, SOURCE: ACS OMEGA, VOLUME: 3, ISSUE: 12
INDEXED IN: Scopus WOS CrossRef: 8
8
TITLE: Clickable 4-Oxo--lactam-Based Selective Probing for Human Neutrophil Elastase Related Proteomes  Full Text
AUTHORS: Eduardo F P Ruivo; Lidia M Goncalves; Luis A R Carvalho; Rita C Guedes; Stefan Hofbauer; Jose A Brito; Margarida Archer; Rui Moreira; Susana D Lucas;
PUBLISHED: 2016, SOURCE: CHEMMEDCHEM, VOLUME: 11, ISSUE: 18
INDEXED IN: Scopus WOS
9
TITLE: Activity-based probes as molecular tools for biomarker discovery
AUTHORS: Carvalho, LAR; Ruivo, EFP; Lucas, SD; Moreira, R;
PUBLISHED: 2015, SOURCE: MEDCHEMCOMM, VOLUME: 6, ISSUE: 4
INDEXED IN: Scopus WOS CrossRef
10
TITLE: A unified approach toward the rational design of selective low nanomolar human neutrophil elastase inhibitors
AUTHORS: Areias, LRP; Ruivo, EFP; Goncalves, LM; Duarte, MT; Andre, V; Moreira, R; Lucas, SD; Guedes, RC;
PUBLISHED: 2015, SOURCE: RSC ADVANCES, VOLUME: 5, ISSUE: 64
INDEXED IN: Scopus WOS CrossRef
IN MY: ORCID
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