Tiago Miguel Guerra Miranda Bandeiras
AuthID: R-000-H93
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TITLE: MoA Studies of the TEAD P-Site Binding Ligand MSC-4106 and Its Optimization to TEAD1-Selective Amide M3686 Full Text
AUTHORS: Heinrich, Timo; Schwarz, Daniel; Petersson, Carl; Gunera, Jakub; Garg, Sakshi; Schneider, Richard; Keil, Marina; Grimmeisen, Lisa; Unzue Lopez, Andrea; Albers, Lisa; Schlesiger, Sarah; Gambardella, Alessia; Bomke, Joerg; Carswell, Emma; Schilke, Heike; Diehl, Patrizia; Doerfel, Benjamin; Musil, Djordje; Trivier, Elisabeth; Broome, Rebecca; ...More
PUBLISHED: 2024, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY
AUTHORS: Heinrich, Timo; Schwarz, Daniel; Petersson, Carl; Gunera, Jakub; Garg, Sakshi; Schneider, Richard; Keil, Marina; Grimmeisen, Lisa; Unzue Lopez, Andrea; Albers, Lisa; Schlesiger, Sarah; Gambardella, Alessia; Bomke, Joerg; Carswell, Emma; Schilke, Heike; Diehl, Patrizia; Doerfel, Benjamin; Musil, Djordje; Trivier, Elisabeth; Broome, Rebecca; ...More
PUBLISHED: 2024, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY
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TITLE: Extract2Chip-Bypassing Protein Purification in Drug Discovery Using Surface Plasmon Resonance
AUTHORS: Paiva, Ana C. F.; Lemos, Ana R.; Busse, Philipp; Martins, Madalena T.; Silva, Diana O.; Freitas, Micael C.; Santos, Sandra P.; Freire, Filipe; Barrey, Evelyne J.; Manival, Xavier; Koetzner, Lisa; Heinrich, Timo; Wegener, Ansgar; Graedler, Ulrich; Bandeiras, Tiago M.; Schwarz, Daniel; Sousa, Pedro M. F.;
PUBLISHED: 2023, SOURCE: BIOSENSORS-BASEL, VOLUME: 13, ISSUE: 10
AUTHORS: Paiva, Ana C. F.; Lemos, Ana R.; Busse, Philipp; Martins, Madalena T.; Silva, Diana O.; Freitas, Micael C.; Santos, Sandra P.; Freire, Filipe; Barrey, Evelyne J.; Manival, Xavier; Koetzner, Lisa; Heinrich, Timo; Wegener, Ansgar; Graedler, Ulrich; Bandeiras, Tiago M.; Schwarz, Daniel; Sousa, Pedro M. F.;
PUBLISHED: 2023, SOURCE: BIOSENSORS-BASEL, VOLUME: 13, ISSUE: 10
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TITLE: Biophysical and structural characterization of the impacts of MET phosphorylation on tepotinib binding
AUTHORS: Ulrich Grädler; Daniel Schwarz; Ansgar Wegener; Thomas Eichhorn; Tiago Bandeiras; Micael Freitas; Alfred Lammens; Oleg Ganichkin; Martin Augustin; Stefano Minguzzi; Frank Becker; Jörg Bomke;
PUBLISHED: 2023, SOURCE: Journal of Biological Chemistry, VOLUME: 299, ISSUE: 11
AUTHORS: Ulrich Grädler; Daniel Schwarz; Ansgar Wegener; Thomas Eichhorn; Tiago Bandeiras; Micael Freitas; Alfred Lammens; Oleg Ganichkin; Martin Augustin; Stefano Minguzzi; Frank Becker; Jörg Bomke;
PUBLISHED: 2023, SOURCE: Journal of Biological Chemistry, VOLUME: 299, ISSUE: 11
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TITLE: Optimization of TEAD P-Site Binding Fragment Hit into In Vivo Active Lead MSC-4106
AUTHORS: Heinrich, Timo; Peterson, Carl; Schneider, Richard; Garg, Sakshi; Schwarz, Daniel; Gunera, Jakub; Seshire, Anita; Koetzner, Lisa; Schlesiger, Sarah; Musil, Djordje; Schilke, Heike; Doerfel, Benjamin; Diehl, Patrizia; Boepple, Pia; Lemos, Ana R.; Sousa, Pedro M. F.; Freire, Filipe; Bandeiras, Tiago M.; Carswell, Emma; Pearson, Nicholas; ...More
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 65, ISSUE: 13
AUTHORS: Heinrich, Timo; Peterson, Carl; Schneider, Richard; Garg, Sakshi; Schwarz, Daniel; Gunera, Jakub; Seshire, Anita; Koetzner, Lisa; Schlesiger, Sarah; Musil, Djordje; Schilke, Heike; Doerfel, Benjamin; Diehl, Patrizia; Boepple, Pia; Lemos, Ana R.; Sousa, Pedro M. F.; Freire, Filipe; Bandeiras, Tiago M.; Carswell, Emma; Pearson, Nicholas; ...More
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 65, ISSUE: 13
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TITLE: Deciphering cellular and molecular determinants of human DPCD protein in complex with RUVBL1/RUVBL2 AAA-ATPases
AUTHORS: Morais, Raphael Dos Santos; Santo, Paulo E.; Ley, Marie; Schelcher, Cedric; Abel, Yoann; Plassart, Laura; Desligniere, Evolene; Chagot, Marie Eve; Quinternet, Marc; Paiva, Ana C. F.; Hessmann, Steve; Morellet, Nelly; Sousa, Pedro M. F.; Vandermoere, Franck; Bertrand, Edouard; Charpentier, Bruno; Bandeiras, Tiago M.; Plisson Chastang, Celia; Verheggen, Celine; Cianferani, Sarah; ...More
PUBLISHED: 2022, SOURCE: JOURNAL OF MOLECULAR BIOLOGY, VOLUME: 434, ISSUE: 19
AUTHORS: Morais, Raphael Dos Santos; Santo, Paulo E.; Ley, Marie; Schelcher, Cedric; Abel, Yoann; Plassart, Laura; Desligniere, Evolene; Chagot, Marie Eve; Quinternet, Marc; Paiva, Ana C. F.; Hessmann, Steve; Morellet, Nelly; Sousa, Pedro M. F.; Vandermoere, Franck; Bertrand, Edouard; Charpentier, Bruno; Bandeiras, Tiago M.; Plisson Chastang, Celia; Verheggen, Celine; Cianferani, Sarah; ...More
PUBLISHED: 2022, SOURCE: JOURNAL OF MOLECULAR BIOLOGY, VOLUME: 434, ISSUE: 19
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TITLE: NOPCHAP1 is a PAQosome cofactor that helps loading NOP58 on RUVBL1/2 during box C/D snoRNP biogenesis
AUTHORS: Abel, Y; Paiva, ACF; Bizarro, J; Chagot, ME; Santo, PE; Robert, MC; Quinternet, M; Vandermoere, F; Sousa, PMF; Fort, P; Charpentier, B; Manival, X; Bandeiras, TM; Bertrand, E; Verheggen, C;
PUBLISHED: 2021, SOURCE: NUCLEIC ACIDS RESEARCH, VOLUME: 49, ISSUE: 2
AUTHORS: Abel, Y; Paiva, ACF; Bizarro, J; Chagot, ME; Santo, PE; Robert, MC; Quinternet, M; Vandermoere, F; Sousa, PMF; Fort, P; Charpentier, B; Manival, X; Bandeiras, TM; Bertrand, E; Verheggen, C;
PUBLISHED: 2021, SOURCE: NUCLEIC ACIDS RESEARCH, VOLUME: 49, ISSUE: 2
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TITLE: Production of high-quality SARS-CoV-2 antigens: Impact of bioprocess and storage on glycosylation, biophysical attributes, and ELISA serologic tests performance Full Text
AUTHORS: Castro, R; Nobre, LS; Eleuterio, RP; Thomaz, M; Pires, A; Monteiro, SM; Mendes, S; Gomes, RA; Clemente, JJ; Sousa, MFQ; Pinto, F; Silva, AC; Freitas, MC; Lemos, AR; Akpogheneta, O; Kosack, L; Bergman, ML; Duarte, N; Matoso, P; Costa, J; ...More
PUBLISHED: 2021, SOURCE: BIOTECHNOLOGY AND BIOENGINEERING, VOLUME: 118, ISSUE: 6
AUTHORS: Castro, R; Nobre, LS; Eleuterio, RP; Thomaz, M; Pires, A; Monteiro, SM; Mendes, S; Gomes, RA; Clemente, JJ; Sousa, MFQ; Pinto, F; Silva, AC; Freitas, MC; Lemos, AR; Akpogheneta, O; Kosack, L; Bergman, ML; Duarte, N; Matoso, P; Costa, J; ...More
PUBLISHED: 2021, SOURCE: BIOTECHNOLOGY AND BIOENGINEERING, VOLUME: 118, ISSUE: 6
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TITLE: Development of antibodies against the notch ligand Delta-Like-1 by phage display with activity against breast cancer cells
AUTHORS: Sales Dias, J; Ferreira, A; Lamy, M; Domenici, G; Monteiro, SMS; Pires, A; Lemos, AR; Kucheryava, K; Nobre, LS; Sousa, PMF; Bandeiras, TM; Silva, G; Barbas, A;
PUBLISHED: 2021, SOURCE: NEW BIOTECHNOLOGY, VOLUME: 64
AUTHORS: Sales Dias, J; Ferreira, A; Lamy, M; Domenici, G; Monteiro, SMS; Pires, A; Lemos, AR; Kucheryava, K; Nobre, LS; Sousa, PMF; Bandeiras, TM; Silva, G; Barbas, A;
PUBLISHED: 2021, SOURCE: NEW BIOTECHNOLOGY, VOLUME: 64
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TITLE: Development of Dl1.72, a Novel Anti-DLL1 Antibody with Anti-Tumor Efficacy against Estrogen Receptor-Positive Breast Cancer Full Text
AUTHORS: Silva, G; Sales Dias, J; Casal, D; Alves, S; Domenici, G; Barreto, C; Matos, C; Lemos, AR; Matias, AT; Kucheryava, K; Ferreira, A; Moita, MR; Braga, S; Brito, C; Cabral, MG; Casalou, C; Barral, DC; Sousa, PMF; Videira, PA; Bandeiras, TM; ...More
PUBLISHED: 2021, SOURCE: CANCERS, VOLUME: 13, ISSUE: 16
AUTHORS: Silva, G; Sales Dias, J; Casal, D; Alves, S; Domenici, G; Barreto, C; Matos, C; Lemos, AR; Matias, AT; Kucheryava, K; Ferreira, A; Moita, MR; Braga, S; Brito, C; Cabral, MG; Casalou, C; Barral, DC; Sousa, PMF; Videira, PA; Bandeiras, TM; ...More
PUBLISHED: 2021, SOURCE: CANCERS, VOLUME: 13, ISSUE: 16
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TITLE: Structural and biophysical insights into the mode of covalent binding of rationally designed potent BMX inhibitors
AUTHORS: Seixas, JD; Sousa, BB; Marques, MC; Guerreiro, A; Traquete, R; Rodrigues, T; Albuquerque, IS; Sousa, MFQ; Lemos, AR; Sousa, PMF; Bandeiras, TM; Wu, D; Doyle, SK; Robinson, CV; Koehler, AN; Corzana, F; Matias, PM; Bernardes, GJL;
PUBLISHED: 2020, SOURCE: RSC CHEMICAL BIOLOGY, VOLUME: 1, ISSUE: 4
AUTHORS: Seixas, JD; Sousa, BB; Marques, MC; Guerreiro, A; Traquete, R; Rodrigues, T; Albuquerque, IS; Sousa, MFQ; Lemos, AR; Sousa, PMF; Bandeiras, TM; Wu, D; Doyle, SK; Robinson, CV; Koehler, AN; Corzana, F; Matias, PM; Bernardes, GJL;
PUBLISHED: 2020, SOURCE: RSC CHEMICAL BIOLOGY, VOLUME: 1, ISSUE: 4