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TITLE: An engineered cereblon optimized for high-throughput screening and molecular glue discovery
AUTHORS: Bailey, Henry J.; Eisert, Jonathan; Kazi, Rubina; Gerhartz, Jan; Pienkowska, Dominika Ewa; Dressel, Ina; Vollrath, Joshua; Kondratov, Ivan; Matviyuk, Tetiana; Tolmachova, Nataliya; Shah, Varun Jayeshkumar; Giuliani, Giulio; Mosler, Thorsten; Geiger, Thomas M.; Esteves, Ana M.; Santos, Sandra P.; Sousa, Raquel L.; Bandeiras, Tiago M.; Leibrock, Eva Maria; Bauer, Ulrike; Leuthner, Birgitta; Langer, Julian D.; Wegener, Ansgar A.; Nowak, Radosla P.; Sorrel, Fiona J.; Dikic, Ivan; ...More
PUBLISHED: 2025, SOURCE: CELL CHEMICAL BIOLOGY, VOLUME: 32, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef
IN MY: ORCID
2
TITLE: Polo-like kinase 1-inhibitor co-complex structures via the surface-entropy reduction approach and a DARPin-assisted approach
AUTHORS: Eberspaecher, Uwe; Schmitz, Arndt A.; Siemeister, Gerhard; Boemer, Ulf; Bandeiras, Tiago M.; Matias, Pedro M.; Schulze, Volker K.; Hillig, Roman C.;
PUBLISHED: 2025, SOURCE: ACTA CRYSTALLOGRAPHICA SECTION D-STRUCTURAL BIOLOGY, VOLUME: 81, ISSUE: 12
INDEXED IN: WOS CrossRef
IN MY: ORCID
3
TITLE: Pushing the limits of hydrogen/deuterium exchange mass spectrometry to study protein:fragment low affinity interactions
AUTHORS: Malta, Catarina F.; Silva, Diana O.; Gradler, Ulrich; Sousa, Pedro M. F.; Musil, Djordje; Schwarz, Daniel; Bomke, Joerg; Bandeiras, Tiago M.; Bortoluzzi, Alessio;
PUBLISHED: 2025, SOURCE: COMMUNICATIONS CHEMISTRY, VOLUME: 8, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef
IN MY: ORCID
4
TITLE: Phenotypic Hit Identification and Optimization of Novel Pan-TEAD and Subtype-Selective Inhibitors  Full Text
AUTHORS: Timo Heinrich; Alessia Gambardella; Daniel Schwarz; Carl Petersson; Jakub Gunera; Sakshi Garg; Richard Schneider; Marina Keil; Lisa Grimmeisen; Andrea Unzue Lopez; Heike Schilke; Thomas Weitzel; Christian Kolb; Patrizia Diehl; Benjamin Doerfel; Uwe Anlauf; Vivian Reither; Corinna Rettig; Beate Opelt; Andrea Delp; Nicole Wildner; Djordje Musil; Erik Friedrich; Lars Burgdorf; Thomas Fuchss; Lisa Albers; Pedro M F Sousa; Filipe Freire; Tiago M. Bandeiras; Dirk Wienke; ...More
PUBLISHED: 2025, SOURCE: Journal of Medicinal Chemistry, VOLUME: 68, ISSUE: 22
INDEXED IN: CrossRef
IN MY: ORCID
5
TITLE: CHEK2 germline variants identified in familial nonmedullary thyroid cancer lead to impaired protein structure and function
AUTHORS: Pires, Carolina; Marques, Ines J.; Valerio, Mariana; Saramago, Ana; Santo, Paulo E.; Santos, Sandra; Silva, Margarida; Moura, Margarida M.; Matos, Joao; Pereira, Teresa; Cabrera, Rafael; Lousa, Diana; Leite, Valeriano; Bandeiras, Tiago M.; Vicente, Joao B.; Cavaco, Branca M.;
PUBLISHED: 2024, SOURCE: JOURNAL OF BIOLOGICAL CHEMISTRY, VOLUME: 300, ISSUE: 3
INDEXED IN: Scopus WOS CrossRef
IN MY: ORCID
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TITLE: Aldehyde Dehydrogenase 2 (ALDH2): A novel sorafenib target in hepatocellular carcinoma unraveled by the proteome-wide cellular thermal shift assay
AUTHORS: Ferreira, Ines C.; Torrejon, Estefania; Abecasis, Bernardo; Alexandre, Bruno M.; Gomes, Ricardo A.; Verslype, Chris; van Pelt, Jos; Barbas, Ana; Sima, Daniel; Bandeiras, Tiago M.; Bortoluzzi, Alessio; Rebelo, Sofia P.;
PUBLISHED: 2024, SOURCE: SLAS DISCOVERY, VOLUME: 29, ISSUE: 3
INDEXED IN: Scopus WOS CrossRef
IN MY: ORCID
7
TITLE: Denaturing mass photometry for rapid optimization of chemical protein-protein cross-linking reactions
AUTHORS: Gizardin Fredon, Hugo; Santo, Paulo E.; Chagot, Marie Eve; Charpentier, Bruno; Bandeiras, Tiago M.; Manival, Xavier; Hernandez Alba, Oscar; Cianferani, Sarah;
PUBLISHED: 2024, SOURCE: NATURE COMMUNICATIONS, VOLUME: 15, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef
IN MY: ORCID
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TITLE: Identification of novel candidate predisposing genes in familial nonmedullary thyroid carcinoma implicating DNA damage repair pathways  Full Text
AUTHORS: Pires, Carolina; Marques, Ines J.; Saramago, Ana; Moura, Margarida M.; Pojo, Marta; Cabrera, Rafael; Santos, Catarina; Rosario, Francisco; Lousa, Diana; Vicente, Joao B.; Bandeiras, Tiago M.; Teixeira, Manuel R. ; Leite, Valeriano; Cavaco, Branca M.;
PUBLISHED: 2024, SOURCE: INTERNATIONAL JOURNAL OF CANCER, VOLUME: 156, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef
IN MY: ORCID
9
TITLE: On the humanization of VHHs: Prospective case studies, experimental and computational characterization of structural determinants for functionality  Full Text
AUTHORS: Fernandez Quintero, Monica L.; Guarnera, Enrico; Musil, Djordje; Pekar, Lukas; Sellmann, Carolin; Freire, Filipe; Sousa, Raquel L.; Santos, Sandra P.; Freitas, Micael C.; Bandeiras, Tiago M.; Silva, Margarida M. S.; Loeffler, Johannes R.; Ward, Andrew B.; Harwardt, Julia; Zielonka, Stefan; Evers, Andreas;
PUBLISHED: 2024, SOURCE: PROTEIN SCIENCE, VOLUME: 33, ISSUE: 11
INDEXED IN: Scopus WOS CrossRef
IN MY: ORCID
10
TITLE: The HSP90/R2TP Quaternary Chaperone Scaffolds Assembly of the TSC Complex  Full Text
AUTHORS: Abeza, Claire; Busse, Philipp; Paiva, Ana C. F.; Chagot, Marie Eve; Schneider, Justine; Robert, Marie Cecile; Vandermoere, Franck; Schaeffer, Christine; Charpentier, Bruno; Sousa, Pedro M. F.; Bandeiras, Tiago M.; Manival, Xavier; Cianferani, Sarah; Bertrand, Edouard; Verheggen, Celine;
PUBLISHED: 2024, SOURCE: JOURNAL OF MOLECULAR BIOLOGY, VOLUME: 436, ISSUE: 23
INDEXED IN: Scopus WOS CrossRef
IN MY: ORCID
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