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TITLE: Rational Design, Synthesis, and Biological Evaluation of Heterocyclic Quinolones Targeting the Respiratory Chain of Mycobacterium tuberculosis  Full Text
AUTHORS: Hong, WD; Gibbons, PD; Leung, SC; Amewu, R; Stocks, PA; Stachulski, A; Horta, P; Cristiano, MLS ; Shone, AE; Moss, D; Ardrey, A; Sharma, R; Warman, AJ; Bedingfield, PTP; Fisher, NE; Aljayyoussi, G; Mead, S; Caws, M; Berry, NG; Ward, SA; Biagini, GA; O’Neill, PM; Nixon, GL; ...More
PUBLISHED: 2017, SOURCE: Journal of Medicinal Chemistry, VOLUME: 60, ISSUE: 9
INDEXED IN: Scopus CrossRef
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TITLE: Novel Endoperoxide-Based Transmission-Blocking Antimalarials with Liver- and Blood-Schizontocidal Activities
AUTHORS: Daniela Miranda; Rita Capela; Ines S Albuquerque; Patricia Meireles; Isa Paiva; Fatima Nogueira; Richard Amewu; Jiri Gut; Philip J Rosenthal; Rudi Oliveira; Maria M Mota ; Rui Moreira; Francesc Marti; Miguel Prudencio ; Paul M O'Neill; Francisca Lopes;
PUBLISHED: 2014, SOURCE: ACS MEDICINAL CHEMISTRY LETTERS, VOLUME: 5, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef
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TITLE: An Endoperoxide-Based Hybrid Approach to Deliver Falcipain Inhibitors Inside Malaria Parasites  Full Text
AUTHORS: Rudi Oliveira; Ana S Newton; Rita C Guedes; Daniela Miranda; Richard K Amewu; Abhishek Srivastava; Jiri Gut; Philip J Rosenthal; Paul M O'Neill; Stephen A Ward; Francisca Lopes ; Rui Moreira ;
PUBLISHED: 2013, SOURCE: CHEMMEDCHEM, VOLUME: 8, ISSUE: 9
INDEXED IN: Scopus WOS CrossRef
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TITLE: Endoperoxide Carbonyl Falcipain 2/3 Inhibitor Hybrids: Toward Combination Chemotherapy of Malaria through a Single Chemical Entity  Full Text
AUTHORS: Peter Gibbons; Edite Verissimo; Nuna C Araujo ; Victoria Barton; Gemma L Nixon; Richard K Amewu; James Chadwick; Paul A Stocks; Giancarlo A Biagini; Abhishek Srivastava; Philip J Rosenthal; Jiri Gut; Rita C Guedes ; Rui Moreira ; Raman Sharma; Neil Berry; Ludes L S Cristiano ; Alison E Shone; Stephen A Ward; Paul M O'Neill;
PUBLISHED: 2010, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 53, ISSUE: 22
INDEXED IN: Scopus WOS CrossRef