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TITLE: Single Mutation on Trastuzumab Modulates the Stability of Antibody-Drug Conjugates Built Using Acetal-Based Linkers and Thiol-Maleimide Chemistry  Full Text
AUTHORS: Ferhati, Xhenti; Jimenez Moreno, Ester; Hoyt, Emily A.; Salluce, Giulia; Cabeza Cabrerizo, Mar; Navo, Claudio D.; Companon, Ismael; Akkapeddi, Padma; Matos, Maria J. ; Salaverri, Noelia; Garrido, Pablo; Martinez, Alfredo; Laserna, Victor; Murray, Thomas, V; Jimenez Oses, Gonzalo; Ravn, Peter; Bernardes, Goncalo J. L.; Corzana, Francisco;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 12
INDEXED IN: Scopus WOS CrossRef: 6
3
TITLE: Molecular basis for fibroblast growth factor 23 O-glycosylation by GalNAc-T3
AUTHORS: Matilde de las Rivas; Earnest James P Paul Daniel; Yoshiki Narimatsu; Ismael Companon; Kentaro Kato; Pablo Hermosilla; Aurelien Thureau; Laura Ceballos Laita; Helena Coelho; Pau Bernado; Filipa Marcelo; Lars Hansen; Ryota Maeda; Anabel Lostao; Francisco Corzana; Henrik Clausen; Thomas A Gerken; Ramon Hurtado Guerrero;
PUBLISHED: 2020, SOURCE: NATURE CHEMICAL BIOLOGY, VOLUME: 16, ISSUE: 3
INDEXED IN: Scopus WOS
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TITLE: Structural characterization of an unprecedented lectin-like antitumoral anti-MUC1 antibody  Full Text
AUTHORS: Macias Leon, J; Bermejo, IA; Asin, A; Garcia Garcia, A; Companon, I; Jimenez Moreno, E; Coelho, H; Mangini, V; Albuquerque, IS; Marcelo, F; Asensio, JL; Bernardes, GJL; Joshi, HJ; Fiammengo, R; Blixt, O; Hurtado Guerrero, R; Corzana, F;
PUBLISHED: 2020, SOURCE: CHEMICAL COMMUNICATIONS, VOLUME: 56, ISSUE: 96
INDEXED IN: WOS
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TITLE: Efficient and irreversible antibody-cysteine bioconjugation using carbonylacrylic reagents
AUTHORS: Barbara Bernardim; Maria J Matos ; Xhenti Ferhati; Ismael Companon; Ana Guerreiro; Padma Akkapeddi; Antonio C B Burtoloso; Gonzalo Jimenez Oses; Francisco Corzana; Goncalo J L Bernardes;
PUBLISHED: 2019, SOURCE: NATURE PROTOCOLS, VOLUME: 14, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef: 46
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TITLE: Structure-Based Design of Potent Tumor-Associated Antigens: Modulation of Peptide Presentation by Single-Atom O/S or O/Se Substitutions at the Glycosidic Linkage  Full Text
AUTHORS: Ismael Companon; Ana Guerreiro; Vincenzo Mangini; Jorge Castro Lopez; Margarita Escudero Casao; Alberto Avenoza; Jesus H Busto; Sergio Castillon; Jesus Jimenez Barbero; Juan L Asensio; Gonzalo Jimenez Oses; Omar Boutureira; Jesus M Peregrina; Ramon Hurtado Guerrero; Roberto Fiammengo; Goncalo J L Bernardes; Francisco Corzana;
PUBLISHED: 2019, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 141, ISSUE: 9
INDEXED IN: WOS
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TITLE: Quaternization of Vinyl/Alkynyl Pyridine Enables Ultrafast Cysteine-Selective Protein Modification and Charge Modulation  Full Text
AUTHORS: Maria J Matos ; Claudio D Navo; Tuuli Hakala; Xhenti Ferhati; Ana Guerreiro; David Hartmann; Barbara Bernardim; Kadi L Saar; Ismael Companon; Francisco Corzana; Tuomas P J Knowles; Gonzalo Jimenez Oses; Goncalo J L Bernardes;
PUBLISHED: 2019, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, VOLUME: 58, ISSUE: 20
INDEXED IN: Scopus WOS CrossRef: 11
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TITLE: Enhanced Permeability and Binding Activity of Isobutylene-Grafted Peptides  Full Text
AUTHORS: Shuang Sun; Ismael Companon; Nuria Martinez Saez; Joao D Seixas; Omar Boutureira; Francisco Corzana; Goncalo J L Bernardes;
PUBLISHED: 2018, SOURCE: CHEMBIOCHEM, VOLUME: 19, ISSUE: 1
INDEXED IN: WOS
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TITLE: Structural and Mechanistic Insights into the Catalytic-Domain-Mediated Short-Range Glycosylation Preferences of GalNAc-T4
AUTHORS: Matilde de las Rivas; Earnest James Paul Daniel; Helena Coelho; Erandi Lira Navarrete; Lluis Raich; Ismael Companon; Ana Diniz; Laura Lagartera; Jesus Jimenez Barbero; Henrik Clausen; Carme Rovira; Filipa Marcelo; Francisco Corzana; Thomas A Gerken; Ramon Hurtado Guerrero;
PUBLISHED: 2018, SOURCE: ACS CENTRAL SCIENCE, VOLUME: 4, ISSUE: 9
INDEXED IN: Scopus WOS
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TITLE: Oxetane Grafts Installed Site-Selectively on Native Disulfides to Enhance Protein Stability and Activity In Vivo  Full Text
AUTHORS: Nuria Martinez Saez; Shuang Sun; Davide Oldrini; Pietro Sormanni; Omar Boutureira; Filippo Carboni; Ismael Companon; Michael J Deery; Michele Vendruscolo; Francisco Corzana; Roberto Adamo; Goncalo J L Bernardes;
PUBLISHED: 2017, SOURCE: ANGEWANDTE CHEMIE-INTERNATIONAL EDITION, VOLUME: 56, ISSUE: 47
INDEXED IN: WOS
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