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TITLE: Elucidating the path to Plasmodium prolyl-tRNA synthetase inhibitors that overcome halofuginone resistance
AUTHORS: Tye, Mark A.; Payne, N. Connor; Johansson, Catrine; Singh, Kritika; Santos, Sofia A.; Fagbami, Lola; Pant, Akansha; Sylvester, Kayla; Luth, Madeline R.; Marques, Sofia; Whitman, Malcolm; Mota, Maria M.; Winzeler, Elizabeth A.; Lukens, Amanda K.; Derbyshire, Emily R.; Oppermann, Udo; Wirth, Dyann F.; Mazitschek, Ralph;
PUBLISHED: 2022, SOURCE: NATURE COMMUNICATIONS, VOLUME: 13, ISSUE: 1
INDEXED IN: Scopus WOS
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TITLE: malERA: An updated research agenda for basic science and enabling technologies in malaria elimination and eradication  Full Text
AUTHORS: Dyann F Wirth; Elizabeth A Winzeler; Fenton, B; John H Adams; Frederic Ariey; Carolina V Barillas Mury; Jake Baum; Sangeeta N Bhatia; Oliver Billker; Selina E Bopp; Flaminia Catteruccia; Alan F Cowman; Chetan E Chitnis; Brendan S Crabb; Kirk W Deitsch; Hernando A Del Portillo; Abdoulaye A Djimde; Carlota Dobano; Patrick E Duffy; Manoj T Duraisingh; Christian Happi; Anthony A James; Gregory LaMonte; Amanda K Lukens; Manuel Llinas; Prashant Mali; Matthias Marti; Jesus Martinez Barnetche; Victoria McGovern; Maria M Mota; Ivo Mueller; Daouda Ndiaye; Daniel E Neafsey; Francine Ntoumi; Jetsumon Prachumsri; Pushkar Sharma; Robert R Shaw; Photini Sinnis; Niraj H Tolia; Sarah K Volkman; Edward A Wenger; Kim Williamson; ...More
PUBLISHED: 2017, SOURCE: PLOS MEDICINE, VOLUME: 14, ISSUE: 11
INDEXED IN: WOS
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TITLE: Exploring the 3-piperidin-4-yl-1H-indole scaffold as a novel antimalarial chemotype  Full Text
AUTHORS: Sofia A Santos; Amanda K Lukens; Lis Coelho; Fatima Nogueira; Dyann F Wirth; Ralph Mazitschek; Rui Moreira; Alexandra Paulo;
PUBLISHED: 2015, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 102
INDEXED IN: Scopus WOS CrossRef
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TITLE: Torins are potent antimalarials that block replenishment of Plasmodium liver stage parasitophorous vacuole membrane proteins
AUTHORS: Kirsten K Hanson ; Ana S Ressurreicao; Kathrin Buchholz; Miguel Prudencio ; Jonathan D Herman Ornelas; Maria Rebelo; Wandy L Beatty; Dyann F Wirth; Thomas Haenscheid; Rui Moreira ; Matthias Marti; Maria M Mota ;
PUBLISHED: 2013, SOURCE: PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, VOLUME: 110, ISSUE: 30
INDEXED IN: Scopus WOS CrossRef