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TITLE: Structure-Based Optimization of Coumarin hA(3) Adenosine Receptor Antagonists  Full Text
AUTHORS: Matos, MJ ; Vilar, S; Vazquez Rodriguez, S; Kachler, S; Klotz, KN; Buccioni, M; Delogu, G; Santana, L; Uriarte, E; Borges, F ;
PUBLISHED: 2020, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 63, ISSUE: 5
INDEXED IN: Scopus WOS CrossRef: 13
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TITLE: Coumarins and adenosine receptors: New perceptions in structure-affinity relationships  Full Text
AUTHORS: Andre Fonseca; Maria Joao Matos ; Santiago Vilar; Sonja Kachler; Karl Norbert Klotz; Eugenio Uriarte; Fernanda Borges ;
PUBLISHED: 2018, SOURCE: CHEMICAL BIOLOGY & DRUG DESIGN, VOLUME: 91, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef: 5
4
TITLE: Discovery of the first A(1) adenosine receptor ligand based on the chromone scaffold
AUTHORS: Cagide, F ; Reis, J; Gaspar, A ; Chavarria, D ; Kachler, S; Klotz, KN; Gomes, LR; Low, JN; Vilar, S; Hripcsak, G; Borges, F ;
PUBLISHED: 2016, SOURCE: RSC ADVANCES, VOLUME: 6, ISSUE: 52
INDEXED IN: Scopus WOS CrossRef: 4
5
TITLE: Progress in the development of small molecules as new human A(3) adenosine receptor ligands based on the 3-thiophenylcoumarin core
AUTHORS: Matos, MJ ; Vilar, S; Kachler, S; Vazquez Rodriguez, S; Varela, C; Delogu, G; Hripcsak, G; Santana, L; Uriarte, E; N Klotz; Borges, F ;
PUBLISHED: 2016, SOURCE: MEDCHEMCOMM, VOLUME: 7, ISSUE: 5
INDEXED IN: Scopus WOS CrossRef: 4
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TITLE: Navigating in chromone chemical space: discovery of novel and distinct A(3) adenosine receptor ligands
AUTHORS: Cagide, F ; Gaspar, A ; Reis, J; Chavarria, D ; Vilar, S; Hripcsak, G; Uriarte, E; Kachler, S; Klotz, KN; Borges, F ;
PUBLISHED: 2015, SOURCE: RSC ADVANCES, VOLUME: 5, ISSUE: 96
INDEXED IN: Scopus WOS CrossRef: 11
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TITLE: Targeting adenosine receptors with coumarins: synthesis and binding activities of amide and carbamate derivatives  Full Text
AUTHORS: Matos, MJ ; Gaspar, A ; Kachler, S; Klotz, KN; Borges, F ; Santana, L; Uriarte, E;
PUBLISHED: 2013, SOURCE: JOURNAL OF PHARMACY AND PHARMACOLOGY, VOLUME: 65, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef: 12
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TITLE: Chalcone-based derivatives as new scaffolds for hA3 adenosine receptor antagonists. Chalcone derivatives as h A 3 receptors   Full Text
AUTHORS: Saleta Vazquez Rodriguez; Maria J Joao Matos ; Lourdes Santana; Eugenio Uriarte; Fernanda Borges ; Sonja Kachler; Karl Norbert Klotz;
PUBLISHED: 2013, SOURCE: JOURNAL OF PHARMACY AND PHARMACOLOGY, VOLUME: 65, ISSUE: 5
INDEXED IN: Scopus WOS CrossRef: 41
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TITLE: Synthesis and adenosine receptors binding affinities of a series of 3-arylcoumarins. AR binding affinities of 3-arylcoumarins  Full Text
AUTHORS: Maria Joao Matos ; Veronika Hogger; Alexandra Gaspar ; Sonja Kachler; Fernanda Borges ; Eugenio Uriarte; Lourdes Santana; Karl Norbert Klotz;
PUBLISHED: 2013, SOURCE: JOURNAL OF PHARMACY AND PHARMACOLOGY, VOLUME: 65, ISSUE: 11
INDEXED IN: Scopus WOS CrossRef: 16