1
TITLE: High-Throughput Phenotypic Screening and Machine Learning Methods Enabled the Selection of Broad-Spectrum Low-Toxicity Antitrypanosomatidic Agents  Full Text
AUTHORS: Linciano, Pasquale; Quotadamo, Antonio; Luciani, Rosaria; Santucci, Matteo; Zorn, Kimberley M.; Foil, Daniel H.; Lane, Thomas R.; da Silva, Anabela Cordeiro; Santarem, Nuno; Moraes, Carolina B.; Freitas Junior, Lucio; Wittig, Ulrike; Mueller, Wolfgang; Tonelli, Michele; Ferrari, Stefania; Venturelli, Alberto; Gul, Sheraz; Kuzikov, Maria; Ellinger, Bernhard; Reinshagen, Jeanette; Ekins, Sean; Costi, Maria Paola; ...More
PUBLISHED: 2023, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 66, ISSUE: 22
INDEXED IN: Scopus WOS
2
TITLE: Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1  Full Text
AUTHORS: Pöhner, I; Quotadamo, A; Panecka Hofman, J; Luciani, R; Santucci, M; Linciano, P; Landi, G; Di Pisa, F; Dello Iacono, L; Pozzi, C; Mangani, S; Gul, S; Witt, G; Ellinger, B; Kuzikov, M; Santarem, N; Cordeiro Da Silva, A ; Costi, MP; Venturelli, A; Wade, RC;
PUBLISHED: 2022, SOURCE: Journal of Medicinal Chemistry, VOLUME: 65, ISSUE: 13
INDEXED IN: Scopus CrossRef: 2
3
TITLE: Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1  Full Text
AUTHORS: Poehner, Ina; Quotadamo, Antonio; Panecka Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro da Silva, Anabela; Costi, Maria P.; Venturelli, Alberto; Wade, Rebecca C.;
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY
INDEXED IN: WOS
4
TITLE: Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1  Full Text
AUTHORS: Poehner, Ina; Quotadamo, Antonio; Panecka Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro da Silva, Anabela; Costi, Maria P.; Venturelli, Alberto; Wade, Rebecca C.;
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 65, ISSUE: 13
INDEXED IN: WOS
5
TITLE: Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth
AUTHORS: Costantino, Luca; Ferrari, Stefania; Santucci, Matteo; Salo Ahen, Outi M. H.; Carosati, Emanuele; Franchini, Silvia; Lauriola, Angela; Pozzi, Cecilia; Trande, Matteo; Gozzi, Gaia; Saxena, Puneet; Cannazza, Giuseppe; Losi, Lorena; Cardinale, Daniela; Venturelli, Alberto; Quotadamo, Antonio; Linciano, Pasquale; Tagliazucchi, Lorenzo; Moschella, Maria Gaetana; Guerrini, Remo; Pacifico, Salvatore; Luciani, Rosaria; Genovese, Filippo; Henrich, Stefan; Alboni, Silvia; Santarem, Nuno; da Silva Cordeiro, Anabela ; Giovannetti, Elisa; Peters, Godefridus J.; Pinton, Paolo; Rimessi, Alessandro; Cruciani, Gabriele; Stroud, Robert M.; Wade, Rebecca C.; Mangani, Stefano; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola; ...More
PUBLISHED: 2022, SOURCE: ELIFE, VOLUME: 11
INDEXED IN: Scopus WOS CrossRef Unpaywall
6
TITLE: Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform
AUTHORS: Carolina B Moraes; Gesa Witt; Maria Kuzikov; Bernhard Ellinper; Theodora Calogeropoulou; Kyriakos C Prousis; Stefano Mangani; Flavio Di Pisa; Giacomo Landi; Lucia Dello Lacono; Cecilia Pozzi; Lucio H Freitas Junior; Bruno dos Santos Pascoalino; Claudia P Bertolacini; Birte Behrens; Oliver Keminer; Jennifer Leu; Markus Wolf; Jeanette Reinshagen; Anabela Cordeiro da Silva ; Nuno Santarem; Alberto Venturelli; Stephen Wrigley; Deepa Karunakaran; Bethlehem Kebede; Ina Poehner; Wolfgang Mueller; Joanna Panecka Hofman; Rebecca C Wade; Martina Fenske; Joachim Clos; Jose M Maria Alunda; Maria J Jesus Corral; Elisa Uliassi; Maria Laura Bolognesi; Pasquale Linciano; Antonio Quotadamo; Stefania Ferrari; Matteo Santucci; Chiara Borsari; Maria Paola Costi; Sheraz Gul; ...More
PUBLISHED: 2019, SOURCE: SLAS DISCOVERY, VOLUME: 24, ISSUE: 3
INDEXED IN: Scopus WOS CrossRef: 2
7
TITLE: Enhancement of Benzothiazoles as Pteridine Reductase-1 Inhibitors for the Treatment of Trypanosomatidic Infections  Full Text
AUTHORS: Pasquale Linciano; Cecilia Pozzi; Lucia dello Iacono; Flavio di Pisa; Giacomo Landi; Alessio Bonucci; Sheraz Gul; Maria Kuzikov; Bernhard Ellinger; Gesa Witt; Nuno Santarem; Catarina Baptista; Caio Franco; Carolina B Moraes; Wolfgang Mueller; Ulrike Wittig; Rosaria Luciani; Antony Sesenna; Antonio Quotadamo; Stefania Ferrari; Ina Pohner; Anabela Cordeiro da Silva ; Stefano Mangani; Luca Costantino; Maria Paola Costi; ...More
PUBLISHED: 2019, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 62, ISSUE: 8
INDEXED IN: Scopus WOS CrossRef
8
TITLE: Aryl thiosemicarbazones for the treatment of trypanosomatidic infections  Full Text
AUTHORS: Pasquale Linciano; Carolina B Moraes; Laura M Alcantara; Caio H Franco; Bruno Pascoalino; Lucio H Freitas Junior; Sara Macedo; Nuno Santarem; Anabela Cordeiro da Silva ; Sheraz Gul; Gesa Witt; Maria Kuzikov; Bernhard Ellinger; Stefania Ferrari; Rosaria Luciani; Antonio Quotadamo; Luca Costantino; Maria Paola Costi;
PUBLISHED: 2018, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 146
INDEXED IN: Scopus WOS CrossRef: 10
9
TITLE: Scaffolds and Biological Targets Avenue to Fight Against Drug Resistance in Leishmaniasis
AUTHORS: Borsari, C; Quotadamo, A; Ferrari, S; Venturelli, A; Cordeiro da Silva, A ; Santarem, N; Costi, MP;
PUBLISHED: 2018, SOURCE: NEGLECTED DISEASES: EXTENSIVE SPACE FOR MODERN DRUG DISCOVERY, VOLUME: 51
INDEXED IN: Scopus WOS CrossRef: 4