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TITLE: Selective Inhibition of Bruton?s Tyrosine Kinase by a Designed Covalent Ligand Leads to Potent Therapeutic Efficacy in Blood Cancers Relative to Clinically Used Inhibitors
AUTHORS: Sousa, Barbara B.; De Almeida, Catia Rebelo; Barahona, Ana F.; Lopes, Raquel; Martins Logrado, Ana; Cavaco, Marco; Neves, Vera; Carvalho, Luis A. R.; Labao Almeida, Carlos; Coelho, Ana R.; Bento, Marta Leal; Lopes, Ricardo M. R. M.; Oliveira, Bruno L.; Castanho, Miguel A. R. B.; Neumeister, Peter; Deutsch, Alexander; Vladimer, Gregory I.; Krall, Nikolaus; Joao, Cristina; Corzana, Francisco; Seixas, Joao D.; Fior, Rita; Bernardes, Goncalo J. L.; ...More
PUBLISHED: 2022, SOURCE: ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE, VOLUME: 5, ISSUE: 11
INDEXED IN: Scopus WOS
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TITLE: Identification of tetracyclic lactams as NMDA receptor antagonists with potential application in neurological disorders  Full Text
AUTHORS: Margarida Espadinha; Lucia Viejo; Ricardo M R M Lopes; Clara Herrera Arozamena; Elies Molins; Daniel J V A dos Santos; Lidia Goncalves; Maria I Isabel Rodriguez Franco; Cristobal de los Rios; Maria M M Santos;
PUBLISHED: 2020, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 194
INDEXED IN: Scopus WOS
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TITLE: N,O-Iminoboronates: Reversible Iminoboronates with Improved Stability for Cancer Cells Targeted Delivery  Full Text
AUTHORS: Ricardo M R M Lopes; Ana E Ventura; Liana C Silva; Helio Faustino; Pedro M P Gois;
PUBLISHED: 2018, SOURCE: CHEMISTRY-A EUROPEAN JOURNAL, VOLUME: 24, ISSUE: 48
INDEXED IN: WOS