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TITLE: Unexpected rearrangement of ivermectin in the synthesis of new derivatives with trypanocidal and antiplasmodial activities  Full Text
AUTHORS: Sulik, Michal; Fontinha, Diana; Steverding, Dietmar; Sobczak, Szymon; Antoszczak, Michal; Prudencio, Miguel; Huczynski, Adam;
PUBLISHED: 2024, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 263
INDEXED IN: Scopus WOS
2
TITLE: New 4-(N-cinnamoylbutyl)aminoacridines as potential multi-stage antiplasmodial leads  Full Text
AUTHORS: Fonte, Melanie; Fontinha, Diana; Moita, Diana; Cano Prades, Omar; Avalos Padilla, Yunuen; Fernandez Busquets, Xavier; Prudencio, Miguel; Paula Gomes ; Teixeira, Catia ;
PUBLISHED: 2023, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 258
INDEXED IN: Scopus WOS CrossRef
3
TITLE: Conjugated carbon monoxide-releasing molecules have broad-spectrum antimicrobial activity
AUTHORS: Mendes, Sofia S.; Sorg, Moritz; Luis, Claudia Malta; Fontinha, Diana; Francisco, Denise; Moita, Diana; Romao, Carlos C.; Pinho, Mariana G.; Pimentel, Catarina; Prudencio, Miguel; Saraiva, Ligia M.;
PUBLISHED: 2023, SOURCE: FUTURE MEDICINAL CHEMISTRY, VOLUME: 15, ISSUE: 12
INDEXED IN: Scopus WOS
6
TITLE: Synthesis and antiplasmodial activity of regioisomers and epimers of second-generation dual acting ivermectin hybrids  Full Text
AUTHORS: Singh, L; Fontinha, D; Francisco, D; Prudencio, M; Singh, K;
PUBLISHED: 2022, SOURCE: SCIENTIFIC REPORTS, VOLUME: 12, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef
7
TITLE: Synthetic antimicrobial peptides as enhancers of the bacteriolytic action of staphylococcal phage endolysins  Full Text
AUTHORS: Gouveia, A; Pinto, D; Veiga, H; Antunes, W; Pinho, MG; Sao Jose, C;
PUBLISHED: 2022, SOURCE: SCIENTIFIC REPORTS, VOLUME: 12, ISSUE: 1
INDEXED IN: Scopus WOS
8
TITLE: A Histone Deacetylase (HDAC) Inhibitor with Pleiotropic In Vitro Anti-Toxoplasma and Anti-Plasmodium Activities Controls Acute and Chronic Toxoplasma Infection in Mice  Full Text
AUTHORS: Jublot, Delphine; Cavailles, Pierre; Kamche, Salima; Francisco, Denise; Fontinha, Diana; Prudencio, Miguel; Guichou, Jean Francois; Labesse, Gilles; Sereno, Denis; Loeuillet, Corinne;
PUBLISHED: 2022, SOURCE: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, VOLUME: 23, ISSUE: 6
INDEXED IN: Scopus WOS CrossRef
9
TITLE: Discovery of spirooxadiazoline oxindoles with dual-stage antimalarial activity  Full Text
AUTHORS: Lopes, Elizabeth A.; Mestre, Raquel; Fontinha, Diana; Legac, Jenny; Pei, Jinxin, V; Sanches Vaz, Margarida; Mori, Mattia; Lehane, Adele M.; Rosenthal, Philip J.; Prudencio, Miguel; Santos, Maria M. M.;
PUBLISHED: 2022, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 236
INDEXED IN: Scopus WOS CrossRef
10
TITLE: Pre-erythrocytic Activity of M5717 in Monotherapy and Combination in Preclinical Plasmodium Infection Models
AUTHORS: Fontinha, Diana; Arez, Francisca; Gal, Isabella Ramella; Nogueira, Goncalo; Moita, Diana; Baeurle, Tobias Hyun Ho; Brito, Catarina; Spangenberg, Thomas; Alves, Paula M.; Prudencio, Miguel;
PUBLISHED: 2022, SOURCE: ACS INFECTIOUS DISEASES, VOLUME: 8, ISSUE: 4
INDEXED IN: Scopus WOS CrossRef
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