21
TITLE: Multistage Antiplasmodium Activity of Astemizole Analogues and Inhibition of Hemozoin Formation as a Contributor to Their Mode of Action
AUTHORS: Malkeet Kumar; John Okombo; Dickson Mambwe; Dale Taylor; Nina Lawrence; Janette Reader; Mariette van der Watt; Diana Fontinha; Margarida Sanches Vaz; Belinda C Bezuidenhout; Sonja B Lauterbach; Dale Liebenberg; Lyn Marie Birkholtz; Theresa L Coetzer; Miguel Prudencio ; Timothy J Egan; Sergio Wittlin; Kelly Chibale;
PUBLISHED: 2019, SOURCE: ACS INFECTIOUS DISEASES, VOLUME: 5, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef: 1
22
TITLE: Structure-Activity Relationship Studies and Plasmodium Life Cycle Profiling Identifies Pan-Active N-Aryl-3-trifluoromethyl Pyrido[1,2-a]benzimidazoles Which Are Efficacious in an in Vivo Mouse Model of Malaria  Full Text
AUTHORS: Godfrey Mayoka; Mathew Njoroge; John Okombo; Liezl Gibhard; Margarida Sanches Vaz; Diana Fontinha; Lyn Marie Birkholtz; Janette Reader; Mariette van der Watt; Theresa L Coetzer; Sonja Lauterbach; Alisje Churchyard; Belinda Bezuidenhout; Timothy J Egan; Clive Yeates; Sergio Wittlin; Miguel Prudencio ; Kelly Chibale;
PUBLISHED: 2019, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 62, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef
23
TITLE: Synthesis and antiplasmodial evaluation of novel mefloquine-based fumardiamides  Full Text
AUTHORS: Maja Beus; Diana Fontinha; Jana Held; Zrinka Rajic; Miguel Prudencio ; Branka Zorc;
PUBLISHED: 2019, SOURCE: ACTA PHARMACEUTICA, VOLUME: 69, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef
25
TITLE: Primaquine homodimers as potential antiplasmodial and anticancer agents  Full Text
AUTHORS: Kristina Pavic; Barbara Rubinic; Zrinka Rajic; Diana Fontinha; Miguel Prudencio ; Lidija Uzelac; Marijeta Kralj; Jana Held; Branka Zorc;
PUBLISHED: 2019, SOURCE: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, VOLUME: 29, ISSUE: 19
INDEXED IN: Scopus WOS
26
TITLE: Primaquine and Chloroquine Fumardiamides as Promising Antiplasmodial Agents  Full Text
AUTHORS: Maja Beus; Diana Fontinha; Jana Held; Zrinka Rajic; Lidija Uzelac; Marijeta Kralj; Miguel Prudencio ; Branka Zorc;
PUBLISHED: 2019, SOURCE: MOLECULES, VOLUME: 24, ISSUE: 15
INDEXED IN: Scopus WOS CrossRef: 1
27
TITLE: Flexible 3D Cell-Based Platforms for the Discovery and Profiling of Novel Drugs Targeting Plasmodium Hepatic Infection
AUTHORS: Francisca Arez; Sofia P Rebelo; Diana Fontinha; Daniel Simao; Tatiana R Martins; Marta Machado; Christoph Fischli; Claude Oeuvray; Lassina Badolo; Manuel J T Carrondo; Matthias Rottmann; Thomas Spangenberg; Catarina Brito; Beatrice Greco; Miguel Prudencio; Paula M Alves;
PUBLISHED: 2019, SOURCE: ACS INFECTIOUS DISEASES, VOLUME: 5, ISSUE: 11
INDEXED IN: Scopus WOS CrossRef: 1
28
TITLE: Primaquine homodimers as potential antiplasmodial and anticancer agents  Full Text
AUTHORS: Kristina Pavić; Barbara Rubinić; Zrinka Rajić; Diana Fontinha; Miguel Prudêncio; Lidija Uzelac; Marijeta Kralj; Jana Held; Branka Zorc;
PUBLISHED: 2019, SOURCE: Bioorganic & Medicinal Chemistry Letters, VOLUME: 29, ISSUE: 19
INDEXED IN: CrossRef
29
TITLE: Primaquine hybrids as promising antimycobacterial and antimalarial agents  Full Text
AUTHORS: Kristina Pavic; Ivana Perkovic; Sarka Pospisilova; Marta Machado; Diana Fontinha; Miguel Prudencio ; Josef Jampilek; Aidan Coffey; Lorraine Endersen; Hrvoje Rimac; Branka Zorc;
PUBLISHED: 2018, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 143
INDEXED IN: Scopus WOS
30
TITLE: SAHAquines, Novel Hybrids Based on SAHA and Primaquine Motifs, as Potential Cytostatic and Antiplasmodial Agents  Full Text
AUTHORS: Maja Beus; Zrinka Rajic; Dusica Maysinger; Zvonimir Mlinaric; Maja Antunovic; Inga Marijanovic; Diana Fontinha; Miguel Prudencio ; Jana Held; Sureyya Olgen; Branka Zorc;
PUBLISHED: 2018, SOURCE: CHEMISTRYOPEN, VOLUME: 7, ISSUE: 8
INDEXED IN: Scopus WOS CrossRef
Page 3 of 4. Total results: 37.