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TITLE: Extract2Chip-Bypassing Protein Purification in Drug Discovery Using Surface Plasmon Resonance  Full Text
AUTHORS: Paiva, Ana C. F.; Lemos, Ana R.; Busse, Philipp; Martins, Madalena T.; Silva, Diana O.; Freitas, Micael C.; Santos, Sandra P.; Freire, Filipe; Barrey, Evelyne J.; Manival, Xavier; Koetzner, Lisa; Heinrich, Timo; Wegener, Ansgar; Graedler, Ulrich; Bandeiras, Tiago M.; Schwarz, Daniel; Sousa, Pedro M. F.;
PUBLISHED: 2023, SOURCE: BIOSENSORS-BASEL, VOLUME: 13, ISSUE: 10
INDEXED IN: Scopus WOS
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TITLE: Biophysical and structural characterization of the impacts of MET phosphorylation on tepotinib binding
AUTHORS: Ulrich Grädler; Daniel Schwarz; Ansgar Wegener; Thomas Eichhorn; Tiago Bandeiras; Micael Freitas; Alfred Lammens; Oleg Ganichkin; Martin Augustin; Stefano Minguzzi; Frank Becker; Jörg Bomke;
PUBLISHED: 2023, SOURCE: Journal of Biological Chemistry, VOLUME: 299, ISSUE: 11
INDEXED IN: Scopus
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TITLE: Optimization of TEAD P-Site Binding Fragment Hit into In Vivo Active Lead MSC-4106  Full Text
AUTHORS: Heinrich, Timo; Peterson, Carl; Schneider, Richard; Garg, Sakshi; Schwarz, Daniel; Gunera, Jakub; Seshire, Anita; Koetzner, Lisa; Schlesiger, Sarah; Musil, Djordje; Schilke, Heike; Doerfel, Benjamin; Diehl, Patrizia; Boepple, Pia; Lemos, Ana R.; Sousa, Pedro M. F.; Freire, Filipe; Bandeiras, Tiago M.; Carswell, Emma; Pearson, Nicholas; Sirohi, Sameer; Hooker, Mollie; Trivier, Elisabeth; Broome, Rebecca; Balsiger, Alexander; Crowden, Abigail; Dillon, Christian; Wienke, Dirk; ...More
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY
INDEXED IN: Scopus WOS
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TITLE: Deciphering cellular and molecular determinants of human DPCD protein in complex with RUVBL1/RUVBL2 AAA-ATPases  Full Text
AUTHORS: Morais, Raphael Dos Santos; Santo, Paulo E.; Ley, Marie; Schelcher, Cedric; Abel, Yoann; Plassart, Laura; Desligniere, Evolene; Chagot, Marie Eve; Quinternet, Marc; Paiva, Ana C. F.; Hessmann, Steve; Morellet, Nelly; Sousa, Pedro M. F.; Vandermoere, Franck; Bertrand, Edouard; Charpentier, Bruno; Bandeiras, Tiago M.; Plisson Chastang, Celia; Verheggen, Celine; Cianferani, Sarah; Manival, Xavier; ...More
PUBLISHED: 2022, SOURCE: JOURNAL OF MOLECULAR BIOLOGY, VOLUME: 434, ISSUE: 19
INDEXED IN: Scopus WOS
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TITLE: Development of Dl1.72, a Novel Anti-DLL1 Antibody with Anti-Tumor Efficacy against Estrogen Receptor-Positive Breast Cancer  Full Text
AUTHORS: Silva, G; Sales Dias, J; Casal, D; Alves, S; Domenici, G; Barreto, C; Matos, C; Lemos, AR; Matias, AT; Kucheryava, K; Ferreira, A; Moita, MR; Braga, S; Brito, C; Cabral, MG; Casalou, C; Barral, DC; Sousa, PMF; Videira, PA; Bandeiras, TM; Barbas, A; ...More
PUBLISHED: 2021, SOURCE: CANCERS, VOLUME: 13, ISSUE: 16
INDEXED IN: WOS
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TITLE: Screening Pyridine Derivatives against Human Hydrogen Sulfide-synthesizing Enzymes by Orthogonal Methods  Full Text
AUTHORS: Karim Zuhra; Pedro M F Sousa; Giulia Paulini; Ana Rita Lemos; Zenta Kalme; Imants Bisenieks; Egils Bisenieks; Brigita Vigante; Gunars Duburs; Tiago M Bandeiras; Luciano Saso; Alessandro Giuffre; Joao B Vicente;
PUBLISHED: 2019, SOURCE: SCIENTIFIC REPORTS, VOLUME: 9, ISSUE: 1
INDEXED IN: Scopus WOS
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TITLE: Production and characterization of a novel Delta-like 1 functional unit as a tool for Notch pathway activation and generation of a specific antibody
AUTHORS: Andreia Ferreira; Marcia Lamy; Maria Margarida Rocha; Gabriela Silva; Tiago M Bandeiras; Ana Barbas;
PUBLISHED: 2018, SOURCE: PROTEIN EXPRESSION AND PURIFICATION, VOLUME: 146
INDEXED IN: Scopus WOS
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TITLE: X-ray structure of full-length human RuvB-Like 2-mechanistic insights into coupling between ATP binding and mechanical action  Full Text
AUTHORS: Sara T N Silva; Jose A Brito; Rocio Arranz; Carlos Oscar S Sorzano; Christine Ebel; James Doutch; Mark D Tully; Jose Maria Carazo; Jose L Carrascosa; Pedro M Matias; Tiago M Bandeiras;
PUBLISHED: 2018, SOURCE: SCIENTIFIC REPORTS, VOLUME: 8, ISSUE: 1
INDEXED IN: Scopus WOS
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TITLE: Insights into the Structures of Superoxide Reductases from the Symbionts Ignicoccus hospitalis and Nanoarchaeum equitans  Full Text
AUTHORS: Celia V Romao; Pedro M Matias; Cristiana M Sousa; Filipa G Pinho; Ana F Pinto; Miguel Teixeira; Tiago M Bandeiras;
PUBLISHED: 2018, SOURCE: BIOCHEMISTRY, VOLUME: 57, ISSUE: 36
INDEXED IN: WOS
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