Stefano Alcaro
AuthID: R-00F-RRP
1
TITLE: Design, synthesis, biological activity evaluation and structure-activity relationships of new steroidal aromatase inhibitors. The case of C-ring and 713 substituted steroids Full Text
AUTHORS: Roleira, Fernanda M. F.; Costa, Saul C.; Gomes, Ana R.; Varela, Carla L.; Amaral, Cristina; Augusto, Tiago, V; Correia da Silva, Georgina; Romeo, Isabella; Costa, Giosue; Alcaro, Stefano; Teixeira, Natercia; Tavares da Silva, Elisiario J.;
PUBLISHED: 2023, SOURCE: BIOORGANIC CHEMISTRY, VOLUME: 131
AUTHORS: Roleira, Fernanda M. F.; Costa, Saul C.; Gomes, Ana R.; Varela, Carla L.; Amaral, Cristina; Augusto, Tiago, V; Correia da Silva, Georgina; Romeo, Isabella; Costa, Giosue; Alcaro, Stefano; Teixeira, Natercia; Tavares da Silva, Elisiario J.;
PUBLISHED: 2023, SOURCE: BIOORGANIC CHEMISTRY, VOLUME: 131
INDEXED IN: Scopus WOS
2
TITLE: 8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin?s antidepressant profile: Synthesis, biological evaluation and docking studies Full Text
AUTHORS: Matos, Maria J. ; Novo, Paula; Mayan, Lucia; Torres, Iria; Uriarte, Eugenio; Yanez, Matilde; Fontenla, Jose Angel; Ortuso, Francesco; Alcaro, Stefano; Procopio, Francesca; Rodriguez Franco, Maria Isabel; Val, Cristina; Loza, Maria I.; Brea, Jose; Borges, Fernanda ; Vina, Dolores;
PUBLISHED: 2023, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 248
AUTHORS: Matos, Maria J. ; Novo, Paula; Mayan, Lucia; Torres, Iria; Uriarte, Eugenio; Yanez, Matilde; Fontenla, Jose Angel; Ortuso, Francesco; Alcaro, Stefano; Procopio, Francesca; Rodriguez Franco, Maria Isabel; Val, Cristina; Loza, Maria I.; Brea, Jose; Borges, Fernanda ; Vina, Dolores;
PUBLISHED: 2023, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 248
3
TITLE: Molecular Modeling and Experimental Evaluation of Non-Chiral Components of Bergamot Essential Oil with Inhibitory Activity against Human Monoamine Oxidases Full Text
AUTHORS: Catalano, Raffaella; Procopio, Francesca; Chavarria, Daniel ; Benfeito, Sofia ; Alcaro, Stefano; Borges, Fernanda ; Ortuso, Francesco;
PUBLISHED: 2022, SOURCE: MOLECULES, VOLUME: 27, ISSUE: 8
AUTHORS: Catalano, Raffaella; Procopio, Francesca; Chavarria, Daniel ; Benfeito, Sofia ; Alcaro, Stefano; Borges, Fernanda ; Ortuso, Francesco;
PUBLISHED: 2022, SOURCE: MOLECULES, VOLUME: 27, ISSUE: 8
4
TITLE: Evaluation of chromane derivatives: Promising privileged scaffolds for lead discovery within Alzheimer's disease Full Text
AUTHORS: Moutayakine, Amina; Marques, Carolina; Lopez, Oscar; Bagetta, Donatella; Leitzbach, Luisa; Hagenow, Stefanie; Carreiro, Elisabete P.; Stark, Holger; Alcaro, Stefano; Fernandez Bolanos, Jose G.; Burke, Anthony J.;
PUBLISHED: 2022, SOURCE: BIOORGANIC & MEDICINAL CHEMISTRY, VOLUME: 68
AUTHORS: Moutayakine, Amina; Marques, Carolina; Lopez, Oscar; Bagetta, Donatella; Leitzbach, Luisa; Hagenow, Stefanie; Carreiro, Elisabete P.; Stark, Holger; Alcaro, Stefano; Fernandez Bolanos, Jose G.; Burke, Anthony J.;
PUBLISHED: 2022, SOURCE: BIOORGANIC & MEDICINAL CHEMISTRY, VOLUME: 68
INDEXED IN: Scopus WOS
5
TITLE: Design and synthesis of chromone-based monoamine oxidase B inhibitors with improved drug-like properties Full Text
AUTHORS: Reis, Joana; Fernandes, Carlos; Salem, Hoda; Maia, Marta; Tome, Claudia; Benfeito, Sofia ; Teixeira, Jose; Oliveira, Paulo J.; Uriarte, Eugenio; Ortuso, Francesco; Alcaro, Stefano; Bagetta, Donatella; Cagide, Fernando ; Borges, Fernanda ;
PUBLISHED: 2022, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 239
AUTHORS: Reis, Joana; Fernandes, Carlos; Salem, Hoda; Maia, Marta; Tome, Claudia; Benfeito, Sofia ; Teixeira, Jose; Oliveira, Paulo J.; Uriarte, Eugenio; Ortuso, Francesco; Alcaro, Stefano; Bagetta, Donatella; Cagide, Fernando ; Borges, Fernanda ;
PUBLISHED: 2022, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 239
6
TITLE: Riluzole-Rasagiline Hybrids: Toward the Development of Multi-Target-Directed Ligands for Amyotrophic Lateral Sclerosis
AUTHORS: Albertini, Claudia; Salerno, Alessandra; Atzenti, Silvia; Uliassi, Elisa; Massenzio, Francesca; Maruca, Annalisa; Rocca, Roberta; Mecava, Marko; Silva, Filomena S. G.; Mena, Debora; Valente, Pedro; Duarte, Ana, I; Chavarria, Daniel ; Bissaro, Maicol; Moro, Stefano; Federico, Stephanie; Spalluto, Giampiero; Soukup, Ondrej; Borges, Fernanda ; Alcaro, Stefano; ...More
PUBLISHED: 2022, SOURCE: ACS CHEMICAL NEUROSCIENCE, VOLUME: 13, ISSUE: 15
AUTHORS: Albertini, Claudia; Salerno, Alessandra; Atzenti, Silvia; Uliassi, Elisa; Massenzio, Francesca; Maruca, Annalisa; Rocca, Roberta; Mecava, Marko; Silva, Filomena S. G.; Mena, Debora; Valente, Pedro; Duarte, Ana, I; Chavarria, Daniel ; Bissaro, Maicol; Moro, Stefano; Federico, Stephanie; Spalluto, Giampiero; Soukup, Ondrej; Borges, Fernanda ; Alcaro, Stefano; ...More
PUBLISHED: 2022, SOURCE: ACS CHEMICAL NEUROSCIENCE, VOLUME: 13, ISSUE: 15
7
TITLE: 4-Oxoquinolines and monoamine oxidase: When tautomerism matters Full Text
AUTHORS: Mesiti, F; Maruca, A; Silva, V; Rocca, R; Fernandes, C; Remiao, F ; Uriarte, E; Alcaro, S; Gaspar, A ; Borges, F ;
PUBLISHED: 2021, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 213
AUTHORS: Mesiti, F; Maruca, A; Silva, V; Rocca, R; Fernandes, C; Remiao, F ; Uriarte, E; Alcaro, S; Gaspar, A ; Borges, F ;
PUBLISHED: 2021, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 213
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TITLE: Mapping Chromone-3-Phenylcarboxamide Pharmacophore: Quid Est Veritas? Full Text
AUTHORS: Mesiti, F; Gaspar, A ; Chavarria, D ; Maruca, A; Rocca, R; Martins, EG; Barreiro, S; Silva, R; Fernandes, C; Gul, S; Keminer, O; Alcaro, S; Borges, F ;
PUBLISHED: 2021, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 64, ISSUE: 15
AUTHORS: Mesiti, F; Gaspar, A ; Chavarria, D ; Maruca, A; Rocca, R; Martins, EG; Barreiro, S; Silva, R; Fernandes, C; Gul, S; Keminer, O; Alcaro, S; Borges, F ;
PUBLISHED: 2021, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 64, ISSUE: 15
9
TITLE: N-1,2,3-triazole-isatin derivatives for cholinesterase and beta-amyloid aggregation inhibition: A comprehensive bioassay study Full Text
AUTHORS: Carolina S Marques; Oscar Lopez; Donatella Bagetta; Elisabete P Carreiro; Sabrina Petralla; Manuela Bartolini; Matthias Hoffmann; Stefano Alcaro; Barbara Monti; Maria Laura Bolognesi; Michael Decker; Jose G Fernandez Bolanos; Anthony J Burke;
PUBLISHED: 2020, SOURCE: BIOORGANIC CHEMISTRY, VOLUME: 98
AUTHORS: Carolina S Marques; Oscar Lopez; Donatella Bagetta; Elisabete P Carreiro; Sabrina Petralla; Manuela Bartolini; Matthias Hoffmann; Stefano Alcaro; Barbara Monti; Maria Laura Bolognesi; Michael Decker; Jose G Fernandez Bolanos; Anthony J Burke;
PUBLISHED: 2020, SOURCE: BIOORGANIC CHEMISTRY, VOLUME: 98
INDEXED IN: Scopus WOS
10
TITLE: C-6 alpha- vs C-7 alpha-Substituted Steroidal Aromatase Inhibitors: Which Is Better? Synthesis, Biochemical Evaluation, Docking Studies, and Structure-Activity Relationships Full Text
AUTHORS: Fernanda M F Roleira; Carla Varela; Cristina Amaral ; Saul C Costa; Georgina Correia da Silva; Federica Moraca; Giosue Costa; Stefano Alcaro; Natercia A A Teixeira ; Elisiario J T Tavares da Silva;
PUBLISHED: 2019, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 62, ISSUE: 7
AUTHORS: Fernanda M F Roleira; Carla Varela; Cristina Amaral ; Saul C Costa; Georgina Correia da Silva; Federica Moraca; Giosue Costa; Stefano Alcaro; Natercia A A Teixeira ; Elisiario J T Tavares da Silva;
PUBLISHED: 2019, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 62, ISSUE: 7