Jose Brea
AuthID: R-00F-X2V
1
TITLE: 8-Amide and 8-carbamate substitution patterns as modulators of 7-hydroxy-4-methylcoumarin?s antidepressant profile: Synthesis, biological evaluation and docking studies Full Text
AUTHORS: Matos, Maria J. ; Novo, Paula; Mayan, Lucia; Torres, Iria; Uriarte, Eugenio; Yanez, Matilde; Fontenla, Jose Angel; Ortuso, Francesco; Alcaro, Stefano; Procopio, Francesca; Rodriguez Franco, Maria Isabel; Val, Cristina; Loza, Maria I.; Brea, Jose; Borges, Fernanda ; Vina, Dolores;
PUBLISHED: 2023, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 248
AUTHORS: Matos, Maria J. ; Novo, Paula; Mayan, Lucia; Torres, Iria; Uriarte, Eugenio; Yanez, Matilde; Fontenla, Jose Angel; Ortuso, Francesco; Alcaro, Stefano; Procopio, Francesca; Rodriguez Franco, Maria Isabel; Val, Cristina; Loza, Maria I.; Brea, Jose; Borges, Fernanda ; Vina, Dolores;
PUBLISHED: 2023, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 248
2
TITLE: Stapling Amantadine to Melanostatin Neuropeptide: Discovery of Potent Positive Allosteric Modulators of the D2 Receptors
AUTHORS: Silva Reis, Sara C.; Correia, Xavier C.; Costa Almeida, Hugo F.; Pires Lima, Beatriz L.; Maronde, Daiane; Costa, Vera M.; Garcia Mera, Xerardo; Cruz, Luis ; Brea, Jose; Loza, Maria Isabel; Rodriguez Borges, Jose E. ; Sampaio Dias, Ivo E. ;
PUBLISHED: 2023, SOURCE: ACS MEDICINAL CHEMISTRY LETTERS, VOLUME: 14, ISSUE: 12
AUTHORS: Silva Reis, Sara C.; Correia, Xavier C.; Costa Almeida, Hugo F.; Pires Lima, Beatriz L.; Maronde, Daiane; Costa, Vera M.; Garcia Mera, Xerardo; Cruz, Luis ; Brea, Jose; Loza, Maria Isabel; Rodriguez Borges, Jose E. ; Sampaio Dias, Ivo E. ;
PUBLISHED: 2023, SOURCE: ACS MEDICINAL CHEMISTRY LETTERS, VOLUME: 14, ISSUE: 12
3
TITLE: Synthesis, Pharmacological, and Biological Evaluation of 2-FuroylBased MIF-1 Peptidomimetics and the Development of a GeneralPurpose Model for Allosteric Modulators (ALLOPTML)
AUTHORS: Sampaio Dias, IE ; Rodríguez Borges, JE ; Yáñez Pérez, V; Arrasate, S; Llorente, J; Brea, JM; Bediaga, H; Viña, D; Loza, MI; Caamaño, O; García Mera, X; González Díaz, H; Sampaio Dias, IE; García Mera, X; González Díaz, H;
PUBLISHED: 2021, SOURCE: ACS CHEMICAL NEUROSCIENCE, VOLUME: 12, ISSUE: 1
AUTHORS: Sampaio Dias, IE ; Rodríguez Borges, JE ; Yáñez Pérez, V; Arrasate, S; Llorente, J; Brea, JM; Bediaga, H; Viña, D; Loza, MI; Caamaño, O; García Mera, X; González Díaz, H; Sampaio Dias, IE; García Mera, X; González Díaz, H;
PUBLISHED: 2021, SOURCE: ACS CHEMICAL NEUROSCIENCE, VOLUME: 12, ISSUE: 1
4
TITLE: Discovery of New Potent Positive Allosteric Modulators of Dopamine D-2 Receptors: Insights into the Bioisosteric Replacement of Proline to 3-Furoic Acid in the Melanostatin Neuropeptide Full Text
AUTHORS: Sampaio Dias, IE ; Reis Mendes, A; Costa, VM; Garcia Mera, X; Brea, J; Loza, MI; Pires Lima, BL; Alcoholado, C; Algarra, M; Rodriguez Borges, JE ;
PUBLISHED: 2021, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 64, ISSUE: 9
AUTHORS: Sampaio Dias, IE ; Reis Mendes, A; Costa, VM; Garcia Mera, X; Brea, J; Loza, MI; Pires Lima, BL; Alcoholado, C; Algarra, M; Rodriguez Borges, JE ;
PUBLISHED: 2021, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 64, ISSUE: 9
5
TITLE: 2-Aryladenine derivatives as a potent scaffold for A(1), A(3) and dual A(1)/A(3) adenosine receptor antagonists: Synthesis and structure-activity relationships Full Text
AUTHORS: Filipe Areias; Carla Correia; Ashly Rocha; Jose Brea; Marian Castro; Maria I Loza; Fernanda Proenca, MF; Alice Carvalho, MA;
PUBLISHED: 2019, SOURCE: BIOORGANIC & MEDICINAL CHEMISTRY, VOLUME: 27, ISSUE: 16
AUTHORS: Filipe Areias; Carla Correia; Ashly Rocha; Jose Brea; Marian Castro; Maria I Loza; Fernanda Proenca, MF; Alice Carvalho, MA;
PUBLISHED: 2019, SOURCE: BIOORGANIC & MEDICINAL CHEMISTRY, VOLUME: 27, ISSUE: 16
INDEXED IN: 
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Scopus WOS6
TITLE: Synthesis, Pharmacological, and Biological Evaluation of MIF-1 Picolinoyl Peptidomimetics as Positive Allosteric Modulators of D2R
AUTHORS: Ivo E Sampaio Dias ; Sara C Silva Reis; Xerardo Garcia Mera; Jose Brea; Isabel Loza, MI; Carla S Alves ; Manuel Algarra; Jose E Rodriguez Borges ;
PUBLISHED: 2019, SOURCE: ACS CHEMICAL NEUROSCIENCE, VOLUME: 10, ISSUE: 8
AUTHORS: Ivo E Sampaio Dias ; Sara C Silva Reis; Xerardo Garcia Mera; Jose Brea; Isabel Loza, MI; Carla S Alves ; Manuel Algarra; Jose E Rodriguez Borges ;
PUBLISHED: 2019, SOURCE: ACS CHEMICAL NEUROSCIENCE, VOLUME: 10, ISSUE: 8
7
TITLE: Enantiospecific Recognition at the A2B Adenosine Receptor by Alkyl 2-Cyanoimino-4-substituted-6-methyl-1,2,3,4-tetrahydropyrimidine-5-carboxylates Full Text
AUTHORS: Carbajales, C; Azuaje, J; Oliveira, A ; Loza, MI; Brea, J; Cadavid, MI; Masaguer, CF; García Mera, X; Gutiérrez De Terán, H; Sotelo, E;
PUBLISHED: 2017, SOURCE: Journal of Medicinal Chemistry, VOLUME: 60, ISSUE: 8
AUTHORS: Carbajales, C; Azuaje, J; Oliveira, A ; Loza, MI; Brea, J; Cadavid, MI; Masaguer, CF; García Mera, X; Gutiérrez De Terán, H; Sotelo, E;
PUBLISHED: 2017, SOURCE: Journal of Medicinal Chemistry, VOLUME: 60, ISSUE: 8
8
TITLE: New chromene scaffolds for adenosine A(2A) receptors: Synthesis, pharmacology and structure-activity relationships Full Text
AUTHORS: Filipe Areias; Marta Costa; Marian Castro; Jose Brea; Elisabet Gregori Puigjane; Fernanda Proenca, MF ; Jordi Mestres; Maria I Loza;
PUBLISHED: 2012, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 54
AUTHORS: Filipe Areias; Marta Costa; Marian Castro; Jose Brea; Elisabet Gregori Puigjane; Fernanda Proenca, MF ; Jordi Mestres; Maria I Loza;
PUBLISHED: 2012, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 54
9
TITLE: Synthesis of novel chromene scaffolds for adenosine receptors Full Text
AUTHORS: Marta Costa; Filipe Areias; Marian Castro; Jose Brea; Maria I Loza; Fernanda Proenca ;
PUBLISHED: 2011, SOURCE: ORGANIC & BIOMOLECULAR CHEMISTRY, VOLUME: 9, ISSUE: 11
AUTHORS: Marta Costa; Filipe Areias; Marian Castro; Jose Brea; Maria I Loza; Fernanda Proenca ;
PUBLISHED: 2011, SOURCE: ORGANIC & BIOMOLECULAR CHEMISTRY, VOLUME: 9, ISSUE: 11
10
TITLE: Synthesis and pharmacological evaluation of novel substituted 9-deazaxanthines as A(2B) receptor antagonists Full Text
AUTHORS: Maria I Isabel Nieto; Maria C Carmen Balo; Jose Brea; Olga Caamano; Franco Fernandez; Xerardo Garcia Mera; Carmen Lopez; Maria I Isabel Loza; Jose Enrique Rodriguez Borges ; Bernat Vidal;
PUBLISHED: 2010, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 45, ISSUE: 7
AUTHORS: Maria I Isabel Nieto; Maria C Carmen Balo; Jose Brea; Olga Caamano; Franco Fernandez; Xerardo Garcia Mera; Carmen Lopez; Maria I Isabel Loza; Jose Enrique Rodriguez Borges ; Bernat Vidal;
PUBLISHED: 2010, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 45, ISSUE: 7
