11
TITLE: A Hybrid of Amodiaquine and Primaquine Linked by Gold(I) Is a Multistage Antimalarial Agent Targeting Heme Detoxification and Thiol Redox Homeostasis  Full Text
AUTHORS: Pereira, Caroline De Souza; Quadros, Helenita Costa; Aboagye, Samuel Yaw; Fontinha, Diana; D'Alessandro, Sarah; Byrne, Margaret Elizabeth; Gendrot, Mathieu; Fonta, Isabelle; Mosnier, Joel; Moreira, Diogo Rodrigo M.; Basilico, Nicoletta; Williams, David. L. L.; Prudencio, Miguel; Pradines, Bruno; Navarro, Maribel;
PUBLISHED: 2022, SOURCE: PHARMACEUTICS, VOLUME: 14, ISSUE: 6
INDEXED IN: Scopus WOS CrossRef
12
TITLE: Broad Spectrum Functional Activity of Structurally Related Monoanionic Au(III) Bis(Dithiolene) Complexes  Full Text
AUTHORS: Le Gal, Yann; Filatre Furcate, Agathe; Lorcy, Dominique; Jeannin, Olivier; Roisnel, Thierry; Dorcet, Vincent; Fontinha, Diana; Francisco, Denise; Prudencio, Miguel; Martins, Marta; Soeiro, Catarina; Sousa, Silvia A.; Leitao, Jorge H.; Morais, Tania S.; Bartolo, Ines; Taveira, Nuno; Guerreiro, Joana F.; Marques, Fernanda;
PUBLISHED: 2022, SOURCE: INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES, VOLUME: 23, ISSUE: 13
INDEXED IN: Scopus WOS CrossRef
14
TITLE: Spiro-beta-lactam BSS-730A Displays Potent Activity against HIV and Plasmodium
AUTHORS: Bartolo, I; Santos, BS; Fontinha, D; Machado, M; Francisco, D; Sepodes, B; Rocha, J; Mota Filipe, H; Pinto, R; Figueira, ME; Barroso, H; Nascimento, T; de Matos, APA; Alves, AJS; Alves, NG; Simoes, CJV; Prudencio, M; Melo, TMVDPE; Taveira, N;
PUBLISHED: 2021, SOURCE: ACS INFECTIOUS DISEASES, VOLUME: 7, ISSUE: 2
INDEXED IN: WOS
15
TITLE: Synthesis and structure-activity relationships of new chiral spiro-beta-lactams highly active against HIV-1 and Plasmodium  Full Text
AUTHORS: Alves, NG; Bartolo, I; Alves, AJS; Fontinha, D; Francisco, D; Lopes, SMM; Soares, MIL; Simoes, CJV; Prudencio, M; Taveira, N; Melo, TMVDPE;
PUBLISHED: 2021, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 219
INDEXED IN: Scopus WOS
16
TITLE: Further investigation of harmicines as novel antiplasmodial agents: Synthesis, structure-activity relationship and insight into the mechanism of action  Full Text
AUTHORS: Marinovic, M; Poje, G; Perkovic, I; Fontinha, D; Prudencio, M; Held, J; de Carvalho, LP; Tandaric, T; Vianello, R; Rajic, Z;
PUBLISHED: 2021, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 224
INDEXED IN: WOS
17
TITLE: Studies of Potency and Efficacy of an Optimized Artemisinin-Quinoline Hybrid against Multiple Stages of the Plasmodium Life Cycle  Full Text
AUTHORS: Quadros, HC; Capci, A; Herrmann, L; D'Alessandro, S; Fontinha, D; Azevedo, R; Villarreal, W; Basilico, N; Prudencio, M; Tsogoeva, SB; Moreira, DRM;
PUBLISHED: 2021, SOURCE: PHARMACEUTICALS, VOLUME: 14, ISSUE: 11
INDEXED IN: Scopus WOS CrossRef
19
TITLE: Spiro-Lactams as Novel Antimicrobial Agents
AUTHORS: Americo J S Alves; Nuno G Alves; Catia C Caratao; Margarida I M Esteves; Diana Fontinha; Ines Bartolo; Maria I L Soares; Susana M M Lopes; Miguel Prudencio ; Nuno Taveira; Teresa M V D P E Pinho e Melo;
PUBLISHED: 2020, SOURCE: CURRENT TOPICS IN MEDICINAL CHEMISTRY, VOLUME: 20, ISSUE: 2
INDEXED IN: Scopus WOS CrossRef
20
TITLE: Harmicines - harmine and cinnamic acid hybrids as novel antiplasmodial hits  Full Text
AUTHORS: Ivana Perkovic; Silvana Raic Malic; Diana Fontinha; Miguel Prudencio; Lais Pessanha de Carvalho; Jana Held; Tana Tandaric; Robert Vianello; Branka Zorc; Zrinka Rajic;
PUBLISHED: 2020, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 187
INDEXED IN: WOS
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