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TITLE: Rational Design, Synthesis, and Biological Evaluation of Heterocyclic Quinolones Targeting the Respiratory Chain of Mycobacterium tuberculosis  Full Text
AUTHORS: Hong, WD; Gibbons, PD; Leung, SC; Amewu, R; Stocks, PA; Stachulski, A; Horta, P; Cristiano, MLS ; Shone, AE; Moss, D; Ardrey, A; Sharma, R; Warman, AJ; Bedingfield, PTP; Fisher, NE; Aljayyoussi, G; Mead, S; Caws, M; Berry, NG; Ward, SA; Biagini, GA; O’Neill, PM; Nixon, GL; ...More
PUBLISHED: 2017, SOURCE: Journal of Medicinal Chemistry, VOLUME: 60, ISSUE: 9
INDEXED IN: Scopus CrossRef
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TITLE: Endoperoxide Carbonyl Falcipain 2/3 Inhibitor Hybrids: Toward Combination Chemotherapy of Malaria through a Single Chemical Entity  Full Text
AUTHORS: Peter Gibbons; Edite Verissimo; Nuna C Araujo ; Victoria Barton; Gemma L Nixon; Richard K Amewu; James Chadwick; Paul A Stocks; Giancarlo A Biagini; Abhishek Srivastava; Philip J Rosenthal; Jiri Gut; Rita C Guedes ; Rui Moreira ; Raman Sharma; Neil Berry; Ludes L S Cristiano ; Alison E Shone; Stephen A Ward; Paul M O'Neill;
PUBLISHED: 2010, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 53, ISSUE: 22
INDEXED IN: Scopus WOS CrossRef
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TITLE: Semi-synthetic and synthetic 1,2,4-trioxaquines and 1,2,4-trioxolaquines: synthesis, preliminary SAR and comparison with acridine endoperoxide conjugates  Full Text
AUTHORS: Nuna C P Araujo; Victoria Barton; Michael Jones; Paul A Stocks; Stephen A Ward; Jill Davies; Patrick G Bray; Alison E Shone; Maria L S Cristiano ; Paul M O'Neill;
PUBLISHED: 2009, SOURCE: BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, VOLUME: 19, ISSUE: 7
INDEXED IN: Scopus WOS CrossRef