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TITLE: Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1  Full Text
AUTHORS: Pöhner, I; Quotadamo, A; Panecka Hofman, J; Luciani, R; Santucci, M; Linciano, P; Landi, G; Di Pisa, F; Dello Iacono, L; Pozzi, C; Mangani, S; Gul, S; Witt, G; Ellinger, B; Kuzikov, M; Santarem, N; Cordeiro Da Silva, A ; Costi, MP; Venturelli, A; Wade, RC;
PUBLISHED: 2022, SOURCE: Journal of Medicinal Chemistry, VOLUME: 65, ISSUE: 13
INDEXED IN: Scopus CrossRef: 2
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TITLE: Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1  Full Text
AUTHORS: Poehner, Ina; Quotadamo, Antonio; Panecka Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro da Silva, Anabela; Costi, Maria P.; Venturelli, Alberto; Wade, Rebecca C.;
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY
INDEXED IN: WOS
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TITLE: Multitarget, Selective Compound Design Yields Potent Inhibitors of a Kinetoplastid Pteridine Reductase 1  Full Text
AUTHORS: Poehner, Ina; Quotadamo, Antonio; Panecka Hofman, Joanna; Luciani, Rosaria; Santucci, Matteo; Linciano, Pasquale; Landi, Giacomo; Di Pisa, Flavio; Dello Iacono, Lucia; Pozzi, Cecilia; Mangani, Stefano; Gul, Sheraz; Witt, Gesa; Ellinger, Bernhard; Kuzikov, Maria; Santarem, Nuno; Cordeiro da Silva, Anabela; Costi, Maria P.; Venturelli, Alberto; Wade, Rebecca C.;
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 65, ISSUE: 13
INDEXED IN: WOS
4
TITLE: Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth
AUTHORS: Costantino, Luca; Ferrari, Stefania; Santucci, Matteo; Salo Ahen, Outi M. H.; Carosati, Emanuele; Franchini, Silvia; Lauriola, Angela; Pozzi, Cecilia; Trande, Matteo; Gozzi, Gaia; Saxena, Puneet; Cannazza, Giuseppe; Losi, Lorena; Cardinale, Daniela; Venturelli, Alberto; Quotadamo, Antonio; Linciano, Pasquale; Tagliazucchi, Lorenzo; Moschella, Maria Gaetana; Guerrini, Remo; Pacifico, Salvatore; Luciani, Rosaria; Genovese, Filippo; Henrich, Stefan; Alboni, Silvia; Santarem, Nuno; da Silva Cordeiro, Anabela ; Giovannetti, Elisa; Peters, Godefridus J.; Pinton, Paolo; Rimessi, Alessandro; Cruciani, Gabriele; Stroud, Robert M.; Wade, Rebecca C.; Mangani, Stefano; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola; ...More
PUBLISHED: 2022, SOURCE: ELIFE, VOLUME: 11
INDEXED IN: Scopus WOS CrossRef Unpaywall
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TITLE: Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-6  Full Text
AUTHORS: Vanden Eynde, JJ; Mangoni, AA; Rautio, J; Leprince, J; Azuma, YT; Garcia Sosa, AT; Hulme, C; Jampilek, J; Karaman, R; Li, W; Paula Gomes ; Hadjipavlou Litina, D; Capasso, R; Geronikaki, A; Cerchia, L; Sabatier, JM; Ragno, R; Tuccinardi, T; Trabocchi, A; Winum, JY; Luque, FJ; Prokai Tatrai, K; Spetea, M; Gutschow, M; Kosalec, I; Guillou, C; Vasconcelos, MH ; Kokotos, G; Rastelli, G; de Sousa, ME ; Manera, C; Gemma, S; Mangani, S; Siciliano, C; Galdiero, S; Liu, H; Scott, PJH; de los Rios, C; Agrofoglio, LA; Collina, S; Guedes, RC; Munoz Torrero, D; ...More
PUBLISHED: 2020, SOURCE: MOLECULES, VOLUME: 25, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef: 2 Unpaywall
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TITLE: Breakthroughs in Medicinal Chemistry: New Targets and Mechanisms, New Drugs, New Hopes-7  Full Text
AUTHORS: Gutschow, M; Vanden Eynde, JJ; Jampilek, J; Kang, CB; Mangoni, AA; Fossa, P; Karaman, R; Trabocchi, A; Scott, PJH; Reynisson, J; Rapposelli, S; Galdiero, S; Winum, JY; Brullo, C; Prokai Tatrai, K; Sharma, AK; Schapira, M; Azuma, YT; Cerchia, L; Spetea, M; Torri, G; Collina, S; Geronikaki, A; Garcia Sosa, AT; Vasconcelos, MH ; Sousa, ME ; Kosalec, I; Tuccinardi, T; Duarte, IF; Salvador, JAR; Bertinaria, M; Pellecchia, M; Amato, J; Rastelli, G; Paula Gomes ; Guedes, RC; Sabatier, JM; Estevez Braun, A; Pagano, B; Mangani, S; Ragno, R; Kokotos, G; Brindisi, M; Gonzalez, FV; Borges, F ; Miloso, M; Rautio, J; Munoz Torrero, D; ...More
PUBLISHED: 2020, SOURCE: MOLECULES, VOLUME: 25, ISSUE: 13
INDEXED IN: Scopus WOS CrossRef: 5 Unpaywall
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TITLE: Accelerating Drug Discovery Efforts for Trypanosomatidic Infections Using an Integrated Transnational Academic Drug Discovery Platform
AUTHORS: Carolina B Moraes; Gesa Witt; Maria Kuzikov; Bernhard Ellinper; Theodora Calogeropoulou; Kyriakos C Prousis; Stefano Mangani; Flavio Di Pisa; Giacomo Landi; Lucia Dello Lacono; Cecilia Pozzi; Lucio H Freitas Junior; Bruno dos Santos Pascoalino; Claudia P Bertolacini; Birte Behrens; Oliver Keminer; Jennifer Leu; Markus Wolf; Jeanette Reinshagen; Anabela Cordeiro da Silva ; Nuno Santarem; Alberto Venturelli; Stephen Wrigley; Deepa Karunakaran; Bethlehem Kebede; Ina Poehner; Wolfgang Mueller; Joanna Panecka Hofman; Rebecca C Wade; Martina Fenske; Joachim Clos; Jose M Maria Alunda; Maria J Jesus Corral; Elisa Uliassi; Maria Laura Bolognesi; Pasquale Linciano; Antonio Quotadamo; Stefania Ferrari; Matteo Santucci; Chiara Borsari; Maria Paola Costi; Sheraz Gul; ...More
PUBLISHED: 2019, SOURCE: SLAS DISCOVERY, VOLUME: 24, ISSUE: 3
INDEXED IN: Scopus WOS CrossRef: 2
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TITLE: Enhancement of Benzothiazoles as Pteridine Reductase-1 Inhibitors for the Treatment of Trypanosomatidic Infections  Full Text
AUTHORS: Pasquale Linciano; Cecilia Pozzi; Lucia dello Iacono; Flavio di Pisa; Giacomo Landi; Alessio Bonucci; Sheraz Gul; Maria Kuzikov; Bernhard Ellinger; Gesa Witt; Nuno Santarem; Catarina Baptista; Caio Franco; Carolina B Moraes; Wolfgang Mueller; Ulrike Wittig; Rosaria Luciani; Antony Sesenna; Antonio Quotadamo; Stefania Ferrari; Ina Pohner; Anabela Cordeiro da Silva ; Stefano Mangani; Luca Costantino; Maria Paola Costi; ...More
PUBLISHED: 2019, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 62, ISSUE: 8
INDEXED IN: Scopus WOS CrossRef
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TITLE: Structural Insights into the Development of Cycloguanil Derivatives as Trypanosoma brucei Pteridine-Reductase-1 Inhibitors
AUTHORS: Giacomo Landi; Pasquale Linciano; Chiara Borsari; Claudia P Bertolacini; Carolina B Moraes; Anabela Cordeiro da Silva ; Sheraz Gul; Gesa Witt; Maria Kuzikov; Maria Paola Costi; Cecilia Pozzi; Stefano Mangani;
PUBLISHED: 2019, SOURCE: ACS INFECTIOUS DISEASES, VOLUME: 5, ISSUE: 7
INDEXED IN: Scopus WOS CrossRef: 1
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TITLE: Chroman-4-One Derivatives Targeting Pteridine Reductase 1 and Showing Anti-Parasitic Activity  Full Text
AUTHORS: Flavio Di Pisa; Giacomo Landi; Lucia Dello Iacono; Cecilia Pozzi; Chiara Borsari; Stefania Ferrari; Matteo Santucci; Nuno Santarem; Anabela Cordeiro da Silva ; Carolina B Moraes; Laura M Alcantara; Vanessa Fontana; Lucio H Freitas Junior; Sheraz Gul; Maria Kuzikov; Birte Behrens; Ina Poehner; Rebecca C Wade; Maria Paola Costi; Stefano Mangani;
PUBLISHED: 2017, SOURCE: MOLECULES, VOLUME: 22, ISSUE: 3
INDEXED IN: Scopus WOS CrossRef
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