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TITLE: Extract2Chip-Bypassing Protein Purification in Drug Discovery Using Surface Plasmon Resonance  Full Text
AUTHORS: Paiva, Ana C. F.; Lemos, Ana R.; Busse, Philipp; Martins, Madalena T.; Silva, Diana O.; Freitas, Micael C.; Santos, Sandra P.; Freire, Filipe; Barrey, Evelyne J.; Manival, Xavier; Koetzner, Lisa; Heinrich, Timo; Wegener, Ansgar; Graedler, Ulrich; Bandeiras, Tiago M.; Schwarz, Daniel; Sousa, Pedro M. F.;
PUBLISHED: 2023, SOURCE: BIOSENSORS-BASEL, VOLUME: 13, ISSUE: 10
INDEXED IN: Scopus WOS
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TITLE: Biophysical and structural characterization of the impacts of MET phosphorylation on tepotinib binding
AUTHORS: Ulrich Grädler; Daniel Schwarz; Ansgar Wegener; Thomas Eichhorn; Tiago Bandeiras; Micael Freitas; Alfred Lammens; Oleg Ganichkin; Martin Augustin; Stefano Minguzzi; Frank Becker; Jörg Bomke;
PUBLISHED: 2023, SOURCE: Journal of Biological Chemistry, VOLUME: 299, ISSUE: 11
INDEXED IN: Scopus
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TITLE: Optimization of TEAD P-Site Binding Fragment Hit into In Vivo Active Lead MSC-4106  Full Text
AUTHORS: Heinrich, Timo; Peterson, Carl; Schneider, Richard; Garg, Sakshi; Schwarz, Daniel; Gunera, Jakub; Seshire, Anita; Koetzner, Lisa; Schlesiger, Sarah; Musil, Djordje; Schilke, Heike; Doerfel, Benjamin; Diehl, Patrizia; Boepple, Pia; Lemos, Ana R.; Sousa, Pedro M. F.; Freire, Filipe; Bandeiras, Tiago M.; Carswell, Emma; Pearson, Nicholas; Sirohi, Sameer; Hooker, Mollie; Trivier, Elisabeth; Broome, Rebecca; Balsiger, Alexander; Crowden, Abigail; Dillon, Christian; Wienke, Dirk; ...More
PUBLISHED: 2022, SOURCE: JOURNAL OF MEDICINAL CHEMISTRY
INDEXED IN: Scopus WOS
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TITLE: Isomorphic diffuse glioma is a morphologically and molecularly distinct tumour entity with recurrent gene fusions of MYBL1 or MYB and a benign disease course  Full Text
AUTHORS: Annika K Wefers; Damian Stichel; Daniel Schrimpf; Roland Coras; Melanie Pages; Arnault Tauziede Espariat; Pascale Varlet; Daniel Schwarz; Figen Soylemezoglu; Ute Pohl; Jose Pimentel; Jochen Meyer; Ekkehard Hewer; Anna Japp; Abhijit Joshi; David E Reuss; Annekathrin Reinhardt; Philipp Sievers; Belen B Casalini; Azadeh Ebrahimi; Kristin Huang; Christian Koelsche; Hu Liang Low; Olinda Rebelo; Dina Marnoto; Albert J Becker; Ori Staszewski; Michel Mittelbronn; Martin Hasselblatt; Jens Schittenhelm; Edmund Cheesman; Ricardo Santos de Oliveira; Rosane Gomes P Queiroz; Elvis Terci Valera; Volkmar H Hans; Andrey Korshunov; Adriana Olar; Keith L Ligon; Stefan M Pfister; Zane Jaunmuktane; Sebastian Brandner; Ruth G Tatevossian; David W Ellison; Thomas S Jacques; Mrinalini Honavar; Eleonora Aronica; Maria Thom; Felix Sahm; Andreas von Deimling; David T W Jones; Ingmar Blumcke; David Capper; ...More
PUBLISHED: 2020, SOURCE: ACTA NEUROPATHOLOGICA, VOLUME: 139, ISSUE: 1
INDEXED IN: Scopus WOS