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TITLE: Single Mutation on Trastuzumab Modulates the Stability of Antibody-Drug Conjugates Built Using Acetal-Based Linkers and Thiol-Maleimide Chemistry  Full Text
AUTHORS: Ferhati, Xhenti; Jimenez Moreno, Ester; Hoyt, Emily A.; Salluce, Giulia; Cabeza Cabrerizo, Mar; Navo, Claudio D.; Companon, Ismael; Akkapeddi, Padma; Matos, Maria J. ; Salaverri, Noelia; Garrido, Pablo; Martinez, Alfredo; Laserna, Victor; Murray, Thomas, V; Jimenez Oses, Gonzalo; Ravn, Peter; Bernardes, Goncalo J. L.; Corzana, Francisco;
PUBLISHED: 2022, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 144, ISSUE: 12
INDEXED IN: Scopus WOS CrossRef: 6
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TITLE: NRARP displays either pro- or anti-tumoral roles in T-cell acute lymphoblastic leukemia depending on Notch and Wnt signaling
AUTHORS: Ines Pinto; Mafalda Duque; Joana Goncalves; Padma Akkapeddi; Mariana L Oliveira; Rita Cabrita; Andres A Yunes; Scott K Durum; Joao T Barata; Rita Fragoso;
PUBLISHED: 2020, SOURCE: ONCOGENE, VOLUME: 39, ISSUE: 5
INDEXED IN: Scopus WOS
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TITLE: Efficient and irreversible antibody-cysteine bioconjugation using carbonylacrylic reagents
AUTHORS: Barbara Bernardim; Maria J Matos ; Xhenti Ferhati; Ismael Companon; Ana Guerreiro; Padma Akkapeddi; Antonio C B Burtoloso; Gonzalo Jimenez Oses; Francisco Corzana; Goncalo J L Bernardes;
PUBLISHED: 2019, SOURCE: NATURE PROTOCOLS, VOLUME: 14, ISSUE: 1
INDEXED IN: Scopus WOS CrossRef: 46
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TITLE: One-pot stapling of interchain disulfides of antibodies using an isobutylene motif  Full Text
AUTHORS: Shuang Sun; Padma Akkapeddi; Marta C Marques; Nuria Martinez Saez; Vukosava M Torres; Carlos Cordeiro; Omar Boutureira; Goncalo J L Bernardes;
PUBLISHED: 2019, SOURCE: ORGANIC & BIOMOLECULAR CHEMISTRY, VOLUME: 17, ISSUE: 7
INDEXED IN: WOS
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TITLE: A fully human anti-IL-7Rα antibody promotes antitumor activity against T-cell acute lymphoblastic leukemia
AUTHORS: Akkapeddi, P; Fragoso, R; Hixon, JA; Ramalho, AS; Oliveira, ML; Carvalho, T; Gloger, A; Matasci, M; Corzana, F; Durum, SK; Neri, D; Bernardes, GJL; Barata, JT;
PUBLISHED: 2019, SOURCE: Leukemia
INDEXED IN: Scopus
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TITLE: Machine intelligence decrypts -lapachone as an allosteric 5-lipoxygenase inhibitor
AUTHORS: Tiago Rodrigues; Markus Werner; Jakob Roth; Eduardo H G da Cruz; Marta C Marques; Padma Akkapeddi; Susana A Lobo; Andreas Koeberle; Francisco Corzana; Eufranio N da Silva Junior; Oliver Werz; Goncalo J L Bernardes;
PUBLISHED: 2018, SOURCE: CHEMICAL SCIENCE, VOLUME: 9, ISSUE: 34
INDEXED IN: Scopus WOS
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TITLE: IL-7R-mediated signaling in T-cell acute lymphoblastic leukemia: An update
AUTHORS: Oliveira, ML; Akkapeddi, P; Ribeiro, D; Melão, A; Barata, JT;
PUBLISHED: 2018, SOURCE: Advances in Biological Regulation
INDEXED IN: Scopus
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TITLE: A Phage Display-Generated Fully Human Anti-IL-7R alpha Antibody Shows Anti-Tumor Activity Against T-Cell Acute Lymphoblastic Leukemia
AUTHORS: Padma Akkapeddi; Ana Rita Fragoso; Julie Hixon; Mariana Oliveira; Tania Carvalho; Andreas Gloger; Mattia Matasci; Francisco Corzana; Scott Durum; Dario Neri; Goncalo Bernardes; Joao Barata;
PUBLISHED: 2018, SOURCE: 60th Annual Meeting of the American-Society-of-Hematology (ASH) in BLOOD, VOLUME: 132
INDEXED IN: WOS
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TITLE: Chemoselective Installation of Amine Bonds on Proteins through Aza-Michael Ligation  Full Text
AUTHORS: Allyson M Freedy; Maria J Matos ; Omar Boutureira; Francisco Corzana; Ana Guerreiro; Padma Akkapeddi; Victor J Somovilla; Tiago Rodrigues; Karl Nicholls; Bangwen Xie; Gonzalo Jimenez Oses; Kevin M Brindle; Andre A Neves; Goncalo J L Bernardes;
PUBLISHED: 2017, SOURCE: JOURNAL OF THE AMERICAN CHEMICAL SOCIETY, VOLUME: 139, ISSUE: 50
INDEXED IN: Scopus WOS CrossRef: 72
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