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TITLE: Destabilizers of the thymidylate synthase homodimer accelerate its proteasomal degradation and inhibit cancer growth
AUTHORS: Costantino, Luca; Ferrari, Stefania; Santucci, Matteo; Salo Ahen, Outi M. H.; Carosati, Emanuele; Franchini, Silvia; Lauriola, Angela; Pozzi, Cecilia; Trande, Matteo; Gozzi, Gaia; Saxena, Puneet; Cannazza, Giuseppe; Losi, Lorena; Cardinale, Daniela; Venturelli, Alberto; Quotadamo, Antonio; Linciano, Pasquale; Tagliazucchi, Lorenzo; Moschella, Maria Gaetana; Guerrini, Remo; Pacifico, Salvatore; Luciani, Rosaria; Genovese, Filippo; Henrich, Stefan; Alboni, Silvia; Santarem, Nuno; da Silva Cordeiro, Anabela ; Giovannetti, Elisa; Peters, Godefridus J.; Pinton, Paolo; Rimessi, Alessandro; Cruciani, Gabriele; Stroud, Robert M.; Wade, Rebecca C.; Mangani, Stefano; Marverti, Gaetano; D'Arca, Domenico; Ponterini, Glauco; Costi, Maria Paola; ...More
PUBLISHED: 2022, SOURCE: ELIFE, VOLUME: 11
INDEXED IN: Scopus WOS CrossRef Unpaywall
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TITLE: SAR Studies and Biological Characterization of a Chromen-4-one Derivative as an Anti-Trypanosoma brucei Agent
AUTHORS: Chiara Borsari; Nuno Santarem; Sara Macedo; Maria D Dolores Jimenez Anton; Juan J Torrado; Ana I Isabel Olias Molero; Maria J Corral; Annalisa Tait; Stefania Ferrari; Luca Costantino; Rosaria Luciani; Glauco Ponterini; Sheraz Gul; Maria Kuzikov; Bernhard Ellinger; Birte Behrens; Jeanette Reinshagen; Jose M Maria Alunda; Anabela Cordeiro da Silva ; Maria Paola Costi;
PUBLISHED: 2019, SOURCE: ACS MEDICINAL CHEMISTRY LETTERS, VOLUME: 10, ISSUE: 4
INDEXED IN: Scopus WOS CrossRef: 1
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TITLE: Discovery of a benzothiophene-flavonol halting miltefosine and antimonial drug resistance in Leishmania parasites through the application of medicinal chemistry, screening and genomics  Full Text
AUTHORS: Chiara Borsari; Maria D Dolores Jimenez Anton; Julia Eick; Eugenia Bifeld; Juan J Jose Torrado; Ana I Isabel Olias Molero; Maria J Jesus Corral; Nuno Santarem; Catarina Baptista; Leda Severi; Sheraz Gul; Markus Wolf; Maria Kuzikov; Bernhard Ellinger; Jeanette Reinshagen; Gesa Witt; Pasquale Linciano; Annalisa Tait; Luca Costantino; Rosaria Luciani; Paloma Tejera Nevado; Dorothea Zander Dinse; Caio H Franco; Stefania Ferrari; Carolina B Moraes; Anabela Cordeiro da Silva ; Glauco Ponterini; Joachim Clos; Jose M Maria Alunda; Maria P Paola Costi; ...More
PUBLISHED: 2019, SOURCE: EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, VOLUME: 183
INDEXED IN: Scopus WOS CrossRef: 1